| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4283367 | 19 | IC50 | = | 6 | uM | ALA5237932 | 5.22 | nM | Homo sapiens | ||
| 2. | ALA4283367 | 19 | FC | = | 3.1 | ALA5237931 | Homo sapiens | |||||
| 3. | ALA4283367 | 19 | EC50 | = | 4 | nM | ALA5237930 | 8.40 | nM | Homo sapiens | ||
| 4. | ALA4283367 | 19 | EC50 | = | 5 | nM | ALA4382894 | 8.30 | nM | |||
| 5. | ALA4283367 | 19 | Activity | 0 | ALA4260947 | Active | Mus musculus | |||||
| 6. | ALA4283367 | 19 | PPB | = | 90 | % | ALA4260945 | % | ||||
| 7. | ALA4283367 | 19 | Drug uptake | = | 0.058 | uM | ALA4260944 | uM | ||||
| 8. | ALA4283367 | 19 | AUC | = | 2.3 | uM.hr | ALA4260943 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 9. | ALA4283367 | 19 | F | = | 53 | % | ALA4260942 | % | Rattus norvegicus | |||
| 10. | ALA4283367 | 19 | CL | = | 22 | ml/min.kg | ALA4260941 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 11. | ALA4283367 | 19 | Ratio | = | 20.2 | ALA4260940 | ||||||
| 12. | ALA4283367 | 19 | log(permeability) | = | -5.4 | ALA4260939 | ||||||
| 13. | ALA4283367 | 19 | IC50 | = | 6 | uM | ALA4260925 | 5.22 | nM | Homo sapiens | ||
| 14. | ALA4283367 | 19 | FC | = | 3.1 | ALA4260920 | ||||||
| 15. | ALA4283367 | 19 | logD | = | 2.92 | ALA4260922 | ||||||
| 16. | ALA4283367 | 19 | EC50 | = | 0.004 | uM | ALA4260921 | 8.40 | nM |
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