| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4284872 | 19 | Emax | = | 74 | % | ALA4251999 | % | Homo sapiens | |||
| 2. | ALA4284872 | 19 | Emax | = | 89 | % | ALA4252017 | % | Homo sapiens | |||
| 3. | ALA4284872 | 19 | Activity | 0 | ALA4251999 | Dose-dependent effect | Homo sapiens | |||||
| 4. | ALA4284872 | 19 | EC50 | > | 25 | uM | ALA4252019 | nM | Homo sapiens | |||
| 5. | ALA4284872 | 19 | EC50 | > | 50 | uM | ALA4252020 | nM | Homo sapiens | |||
| 6. | ALA4284872 | 19 | Kd | = | 0.3 | uM | ALA4252018 | 6.52 | nM | Homo sapiens | ||
| 7. | ALA4284872 | 19 | EC50 | = | 0.6 | uM | ALA4252017 | 6.22 | nM | Homo sapiens | ||
| 8. | ALA4284872 | 19 | FC | = | 1.6 | ALA4252016 | Homo sapiens | |||||
| 9. | ALA4284872 | 19 | FC | = | 2.1 | ALA4252015 | Homo sapiens | |||||
| 10. | ALA4284872 | 19 | FC | = | 2.7 | ALA4252014 | Homo sapiens | |||||
| 11. | ALA4284872 | 19 | FC | = | 4.9 | ALA4252013 | Homo sapiens | |||||
| 12. | ALA4284872 | 19 | FC | = | 6.7 | ALA4252012 | Homo sapiens | |||||
| 13. | ALA4284872 | 19 | t1/2 | = | 1.1 | hr | ALA4252011 | hr | Mus musculus | |||
| 14. | ALA4284872 | 19 | Vdss | = | 1.4 | L/Kg | ALA4252010 | L.kg-1 | Mus musculus | |||
| 15. | ALA4284872 | 19 | CL | = | 2.3 | L/hr/kg | ALA4252009 | mL.min-1.kg-1 | Mus musculus | |||
| 16. | ALA4284872 | 19 | CLH | = | 150 | uL/min.mg | ALA4252004 | mL.min-1.g-1 | ||||
| 17. | ALA4284872 | 19 | solubility | = | 96 | uM | ALA4252003 | nM | ||||
| 18. | ALA4284872 | 19 | Ratio | = | 2.5 | ALA4252002 | ||||||
| 19. | ALA4284872 | 19 | Ratio | = | 1.5 | ALA4252001 | ||||||
| 20. | ALA4284872 | 19 | Papp | = | 39 | ucm/s | ALA4252000 | ucm/s |
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