| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4285743 | A | AUC | = | 434 | ng.hr/ml | ALA4261365 | ng.hr.mL-1 | Mus musculus | |||
| 2. | ALA4285743 | A | Cp | 0 | ALA4261363 | Bld | ||||||
| 3. | ALA4285743 | A | Tmax | = | 2 | hr | ALA4261361 | hr | Mus musculus | |||
| 4. | ALA4285743 | A | Cmax | = | 252 | nM | ALA4261359 | nM | Mus musculus | |||
| 5. | ALA4285743 | A | t1/2 | = | 46 | min | ALA4261358 | hr | ||||
| 6. | ALA4285743 | A | t1/2 | = | 60 | min | ALA4261357 | hr | ||||
| 7. | ALA4285743 | A | solubility | = | 50 | uM | ALA4261356 | nM | ||||
| 8. | ALA4285743 | A | INH | = | 47 | % | ALA4261354 | % | Mus musculus | |||
| 9. | ALA4285743 | A | IC50 | = | 25 | nM | ALA4261351 | 7.60 | nM | Mus musculus | ||
| 10. | ALA4285743 | A | INH | = | 81 | % | ALA4261345 | % | Mus musculus | |||
| 11. | ALA4285743 | A | Ratio IC50 | = | 3 | ALA4261350 | ||||||
| 12. | ALA4285743 | A | IC50 | = | 6 | nM | ALA4261347 | 8.22 | nM | Homo sapiens | ||
| 13. | ALA4285743 | A | IC50 | = | 2 | nM | ALA4261346 | 8.70 | nM | Homo sapiens | ||
| 14. | ALA4285743 | A | t1/2 | = | 60 | min | ALA4400659 | hr | ||||
| 15. | ALA4285743 | A | Activity | 0 | ALA4400692 | Non-Toxic | Mus musculus | |||||
| 16. | ALA4285743 | A | Activity | 0 | ALA4400691 | Non-Toxic | ||||||
| 17. | ALA4285743 | A | Activity | 0 | ALA4400690 | Active | Mus musculus | |||||
| 18. | ALA4285743 | A | Activity | 0 | ALA4400689 | Active | Mus musculus | |||||
| 19. | ALA4285743 | A | Activity | 0 | ALA4400688 | Active | Mus musculus | |||||
| 20. | ALA4285743 | A | FC | = | 2 | ALA4400687 | Mus musculus |
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