# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4289255 | 3; 001 | pIC50 | 0 | ALA4257143 | Not Determined | Homo sapiens | |||||
2. | ALA4289255 | 3; 001 | pIC50 | 0 | ALA4257142 | Not Determined | Homo sapiens | |||||
3. | ALA4289255 | 3; 001 | pIC50 | 0 | ALA4257141 | Not Determined | Rattus norvegicus | |||||
4. | ALA4289255 | 3; 001 | Activity | = | 57 | % | ALA4257115 | % | Rattus norvegicus | |||
5. | ALA4289255 | 3; 001 | Activity | = | 41 | % | ALA4257112 | % | Rattus norvegicus | |||
6. | ALA4289255 | 3; 001 | pIC50 | = | 7.4 | ALA4257109 | 7.40 | nM | Rattus norvegicus | |||
7. | ALA4289255 | 3; 001 | pIC50 | = | 7.4 | ALA4257110 | 7.40 | nM | Homo sapiens | |||
8. | ALA4289255 | 3; 001 | INH | 0 | ALA5149736 | Active | % | |||||
9. | ALA4289255 | 3; 001 | INH | 0 | ALA5149735 | Active | % | |||||
10. | ALA4289255 | 3; 001 | AUC/dose | = | 12 | ng.hr/ml | ALA5149731 | ng.hr/ml | ||||
11. | ALA4289255 | 3; 001 | Cmax | = | 6 | ng/ml | ALA5149730 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
12. | ALA4289255 | 3; 001 | pIC50 | = | 7.4 | ALA5149727 | 7.40 | nM | Rattus norvegicus | |||
13. | ALA4289255 | 3; 001 | pIC50 | = | 7.6 | ALA5149726 | 7.60 | nM | Homo sapiens |