| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4289325 | 13 | Drug metabolism | 0 | ALA4270347 | Metabolite_Notdetected | ||||||
| 2. | ALA4289325 | 13 | Drug metabolism | = | 19 | % | ALA4270345 | % | ||||
| 3. | ALA4289325 | 13 | Stability | = | 81 | % | ALA4270344 | % | ||||
| 4. | ALA4289325 | 13 | Cp | = | 0.47 | uM | ALA4270343 | uM | ||||
| 5. | ALA4289325 | 13 | AUC | = | 31.2 | uM.hr | ALA4270342 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Macaca mulatta | ||
| 6. | ALA4289325 | 13 | Cmax | = | 2.99 | uM | ALA4270339 | nM | Macaca mulatta | |||
| 7. | ALA4289325 | 13 | Cp(f) | = | 0.018 | uM | ALA4270341 | uM | ||||
| 8. | ALA4289325 | 13 | Fu | = | 2.3 | % | ALA4270338 | |||||
| 9. | ALA4289325 | 13 | Activity | = | 65 | % | ALA4270337 | % | Mus musculus | |||
| 10. | ALA4289325 | 13 | t1/2 | = | 1.6 | hr | ALA4270336 | hr | Rattus norvegicus | |||
| 11. | ALA4289325 | 13 | F | = | 85 | % | ALA4270335 | % | Rattus norvegicus | |||
| 12. | ALA4289325 | 13 | AUC | = | 8.5 | uM.hr | ALA4270334 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 13. | ALA4289325 | 13 | CL | = | 3.4 | ml/min.kg | ALA4270333 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 14. | ALA4289325 | 13 | Activity | 0 | ALA4270332 | Not Active | Homo sapiens | |||||
| 15. | ALA4289325 | 13 | INH | 0 | ALA4270331 | Not Active | % | Homo sapiens | ||||
| 16. | ALA4289325 | 13 | INH | 0 | ALA4270330 | Not Active | % | Homo sapiens | ||||
| 17. | ALA4289325 | 13 | INH | 0 | ALA4270329 | Not Active | % | Homo sapiens | ||||
| 18. | ALA4289325 | 13 | IC50 | > | 10 | uM | ALA4270328 | nM | Homo sapiens | |||
| 19. | ALA4289325 | 13 | IC50 | > | 10 | uM | ALA4270327 | nM | Homo sapiens | |||
| 20. | ALA4289325 | 13 | IC50 | > | 10 | uM | ALA4270326 | nM | Homo sapiens |
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