# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4291464 | R-C025 | Drug uptake | 0 | ALA4256888 | Active | ||||||
2. | ALA4291464 | R-C025 | Drug metabolism | 0 | ALA4256885 | Metabolite_Detected | ||||||
3. | ALA4291464 | R-C025 | Cp | > | 20 | uM | ALA4256883 | uM | ||||
4. | ALA4291464 | R-C025 | AUC | = | 1081 | nmol.hr/ml | ALA4256876 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Macaca fascicularis | ||
5. | ALA4291464 | R-C025 | t1/2 | = | 9.3 | hr | ALA4256870 | hr | Macaca fascicularis | |||
6. | ALA4291464 | R-C025 | Cmax | = | 79 | uM | ALA4256864 | nM | Macaca fascicularis | |||
7. | ALA4291464 | R-C025 | Tmax | = | 2.5 | hr | ALA4256858 | hr | Macaca fascicularis | |||
8. | ALA4291464 | R-C025 | IC50 | = | 23 | nM | ALA4256853 | 7.64 | nM | Homo sapiens |