# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4299371 | 3; AKG115 | Activity | 0 | ALA3738467 | Toxic | Rattus norvegicus | |||||
2. | ALA4299371 | 3; AKG115 | Activity | = | 24 | % | ALA3738466 | % | Rattus norvegicus | |||
3. | ALA4299371 | 3; AKG115 | Stability | = | 75 | % | ALA3738464 | % | Rattus norvegicus | |||
4. | ALA4299371 | 3; AKG115 | Stability | = | 78 | % | ALA3738463 | % | Rattus norvegicus | |||
5. | ALA4299371 | 3; AKG115 | Stability | = | 82 | % | ALA3738462 | % | Rattus norvegicus | |||
6. | ALA4299371 | 3; AKG115 | Stability | = | 87 | % | ALA3738461 | % | Rattus norvegicus | |||
7. | ALA4299371 | 3; AKG115 | Stability | = | 90 | % | ALA3738460 | % | Rattus norvegicus | |||
8. | ALA4299371 | 3; AKG115 | Stability | = | 95 | % | ALA3738459 | % | Rattus norvegicus | |||
9. | ALA4299371 | 3; AKG115 | Stability | = | 100 | % | ALA3738458 | % | Rattus norvegicus | |||
10. | ALA4299371 | 3; AKG115 | Ke | = | 13 | nM | ALA3738457 | nM | Homo sapiens | |||
11. | ALA4299371 | 3; AKG115 | Ratio IC50 | = | 1.3 | ALA3738456 | ||||||
12. | ALA4299371 | 3; AKG115 | IC50 | = | 30 | nM | ALA3738455 | 7.52 | nM | Homo sapiens | ||
13. | ALA4299371 | 3; AKG115 | IC50 | = | 39 | nM | ALA3738454 | 7.41 | nM | Homo sapiens | ||
14. | ALA4299371 | 3; AKG115 | Ke | = | 9.7 | nM | ALA3738452 | nM | Cavia porcellus | |||
15. | ALA4299371 | 3; AKG115 | Activity | 0 | ALA3738450 | Not Active | Cavia porcellus | |||||
16. | ALA4299371 | 3; AKG115 | IC50 | = | 31 | nM | ALA3738447 | 7.51 | nM | Mus musculus | ||
17. | ALA4299371 | 3; AKG115 | pIC50 | = | 7.92 | ALA3738444 | 7.92 | nM | Homo sapiens | |||
18. | ALA4299371 | 3; AKG115 | Ki | = | 5 | nM | ALA3738444 | 8.30 | nM | Homo sapiens | ||
19. | ALA4299371 | 3; AKG115 | pIC50 | = | 8.78 | ALA3738443 | 8.78 | nM | Homo sapiens | |||
20. | ALA4299371 | 3; AKG115 | Ki | = | 1 | nM | ALA3738443 | 9.00 | nM | Homo sapiens |