# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4299479 | 7; AKG190 | Activity | 0 | ALA3738450 | Not Active | Cavia porcellus | |||||
2. | ALA4299479 | 7; AKG190 | t1/2 | > | 2 | hr | ALA3738465 | hr | Rattus norvegicus | |||
3. | ALA4299479 | 7; AKG190 | Ke | = | 5.8 | nM | ALA3738452 | nM | Cavia porcellus | |||
4. | ALA4299479 | 7; AKG190 | Ratio IC50 | = | 5 | ALA3738448 | ||||||
5. | ALA4299479 | 7; AKG190 | IC50 | = | 12 | nM | ALA3738447 | 7.92 | nM | Mus musculus | ||
6. | ALA4299479 | 7; AKG190 | pIC50 | = | 7.81 | ALA3738444 | 7.81 | nM | Homo sapiens | |||
7. | ALA4299479 | 7; AKG190 | Ki | = | 7 | nM | ALA3738444 | 8.15 | nM | Homo sapiens | ||
8. | ALA4299479 | 7; AKG190 | pIC50 | = | 8.08 | ALA3738443 | 8.08 | nM | Homo sapiens | |||
9. | ALA4299479 | 7; AKG190 | Ki | = | 4 | nM | ALA3738443 | 8.40 | nM | Homo sapiens | ||
10. | ALA4299479 | 7; AKG190 | Ki | = | 34 | nM | ALA3738442 | 7.47 | nM | Rattus norvegicus | ||
11. | ALA4299479 | 7; AKG190 | Ki | = | 5.6 | nM | ALA3738441 | 8.25 | nM | Homo sapiens | ||
12. | ALA4299479 | 7; AKG190 | IC50 | = | 65 | nM | ALA3738446 | 7.19 | nM | Cavia porcellus | ||
13. | ALA4299479 | 7; AKG190 | Stability | = | 0.16 | % | ALA3738464 | % | Rattus norvegicus | |||
14. | ALA4299479 | 7; AKG190 | Stability | = | 14 | % | ALA3738463 | % | Rattus norvegicus | |||
15. | ALA4299479 | 7; AKG190 | Stability | = | 28 | % | ALA3738462 | % | Rattus norvegicus | |||
16. | ALA4299479 | 7; AKG190 | Stability | = | 52 | % | ALA3738461 | % | Rattus norvegicus | |||
17. | ALA4299479 | 7; AKG190 | Stability | = | 68 | % | ALA3738460 | % | Rattus norvegicus | |||
18. | ALA4299479 | 7; AKG190 | Stability | = | 84 | % | ALA3738459 | % | Rattus norvegicus | |||
19. | ALA4299479 | 7; AKG190 | Stability | = | 100 | % | ALA3738458 | % | Rattus norvegicus |