| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4299745 | 5 | FC | > | 2 | ALA4149353 | Mycobacterium tuberculosis | |||||
| 2. | ALA4299745 | 5 | FC | = | 5 | ALA4149354 | Mycobacterium tuberculosis | |||||
| 3. | ALA4299745 | 5 | FC | = | 1.5 | ALA4149355 | Mycobacterium tuberculosis | |||||
| 4. | ALA4299745 | 5 | AUC | = | 58 | microg.min/mL | ALA4149356 | ng.hr.mL-1 | Rattus norvegicus | |||
| 5. | ALA4299745 | 5 | AUC | = | 278 | microg.min/mL | ALA4149357 | ng.hr.mL-1 | Rattus norvegicus | |||
| 6. | ALA4299745 | 5 | Vdss | = | 0.57 | L/Kg | ALA4149358 | L.kg-1 | Rattus norvegicus | |||
| 7. | ALA4299745 | 5 | CL | = | 8.9 | ml/min.kg | ALA4149359 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 8. | ALA4299745 | 5 | beta t1/2 | = | 40 | min | ALA4149360 | hr | Rattus norvegicus | |||
| 9. | ALA4299745 | 5 | F | = | 2.1 | % | ALA4149361 | % | Rattus norvegicus | |||
| 10. | ALA4299745 | 5 | CC50 | > | 200 | uM | ALA4149348 | nM | Chlorocebus sabaeus | |||
| 11. | ALA4299745 | 5 | CC50 | > | 200 | uM | ALA4149347 | nM | Homo sapiens | |||
| 12. | ALA4299745 | 5 | MIC99 | = | 2.3 | uM | ALA4149346 | uM | Mycobacterium tuberculosis | |||
| 13. | ALA4299745 | 5 | Ki(app) | = | 11.6 | nM | ALA4149345 | 7.94 | nM | Mycobacterium tuberculosis | ||
| 14. | ALA4299745 | 5 | MIC | >= | 50 | uM | ALA4149350 | nM | Mycobacterium tuberculosis | |||
| 15. | ALA4299745 | 5 | Activity | 0 | ALA4149349 | Not Active | Mycobacterium tuberculosis |
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