# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4436124 | 11b | Drug metabolism | = | 0.3 | % | ALA4322490 | % | Homo sapiens | |||
2. | ALA4436124 | 11b | Stability | = | 99.7 | % | ALA4322520 | % | Homo sapiens | |||
3. | ALA4436124 | 11b | Stability | = | 73.3 | % | ALA4322519 | % | Homo sapiens | |||
4. | ALA4436124 | 11b | Stability | = | 93.2 | % | ALA4322516 | % | ||||
5. | ALA4436124 | 11b | Stability | = | 93 | % | ALA4322515 | % | ||||
6. | ALA4436124 | 11b | Stability | = | 93.6 | % | ALA4322514 | % | ||||
7. | ALA4436124 | 11b | Stability | = | 81.2 | % | ALA4322513 | % | ||||
8. | ALA4436124 | 11b | Selectivity ratio | = | 8.6 | ALA4322510 | ||||||
9. | ALA4436124 | 11b | Kd | = | 980 | nM | ALA4322509 | 6.01 | nM | Homo sapiens | ||
10. | ALA4436124 | 11b | Kd | > | 30000 | nM | ALA4322508 | nM | Homo sapiens | |||
11. | ALA4436124 | 11b | Kd | = | 1800 | nM | ALA4322507 | 5.75 | nM | Homo sapiens | ||
12. | ALA4436124 | 11b | Kd | = | 1900 | nM | ALA4322506 | 5.72 | nM | Homo sapiens | ||
13. | ALA4436124 | 11b | Kd | = | 1400 | nM | ALA4322505 | 5.85 | nM | Homo sapiens | ||
14. | ALA4436124 | 11b | Kd | = | 120 | nM | ALA4322504 | 6.92 | nM | Homo sapiens | ||
15. | ALA4436124 | 11b | Kd | = | 14 | nM | ALA4322503 | 7.85 | nM | Homo sapiens | ||
16. | ALA4436124 | 11b | Stability | = | 91 | % | ALA4322502 | % | Homo sapiens | |||
17. | ALA4436124 | 11b | Stability | = | 93 | % | ALA4322501 | % | Homo sapiens | |||
18. | ALA4436124 | 11b | Stability | = | 73 | % | ALA4322500 | % | Homo sapiens | |||
19. | ALA4436124 | 11b | Stability | = | 51 | % | ALA4322499 | % | Homo sapiens | |||
20. | ALA4436124 | 11b | Ratio Ki | = | 214 | ALA4322498 |