# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4436134 | 4be | Activity | 0 | ALA4375448 | Active | Mus musculus | |||||
2. | ALA4436134 | 4be | Activity | 0 | ALA4375447 | Active | Mus musculus | |||||
3. | ALA4436134 | 4be | Activity | 0 | ALA4375437 | Active | Mus musculus | |||||
4. | ALA4436134 | 4be | F | = | 16 | % | ALA4375425 | % | ||||
5. | ALA4436134 | 4be | AUC | = | 418 | micromol.hr/L | ALA4375430 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
6. | ALA4436134 | 4be | IC50 | = | 0.025 | uM | ALA4375439 | 7.60 | nM | Mus musculus | ||
7. | ALA4436134 | 4be | INH | 0 | ALA4375442 | Not Active | % | Mus musculus | ||||
8. | ALA4436134 | 4be | INH | 0 | ALA4375441 | Not Active | % | Mus musculus | ||||
9. | ALA4436134 | 4be | IC50 | = | 0.023 | uM | ALA4375440 | 7.64 | nM | Mus musculus | ||
10. | ALA4436134 | 4be | AUC | = | 69 | micromol.hr/L | ALA4375432 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
11. | ALA4436134 | 4be | Tmax | = | 0.8 | hr | ALA4375434 | hr | ||||
12. | ALA4436134 | 4be | Tmax | = | 0.8 | hr | ALA4375433 | hr | ||||
13. | ALA4436134 | 4be | Cmax | = | 70.2 | uM | ALA4375436 | nM | ||||
14. | ALA4436134 | 4be | Cmax | = | 12.9 | uM | ALA4375435 | nM | ||||
15. | ALA4436134 | 4be | Drug uptake | 0 | ALA4375445 | Active | ||||||
16. | ALA4436134 | 4be | INH | 0 | ALA4375443 | Not Active | % | Homo sapiens | ||||
17. | ALA4436134 | 4be | F | = | 16.4 | % | ALA5053152 | % | ||||
18. | ALA4436134 | 4be | INH | 0 | ALA5053142 | Active | % | |||||
19. | ALA4436134 | 4be | INH | 0 | ALA5053141 | Active | % | |||||
20. | ALA4436134 | 4be | INH | 0 | ALA5053140 | Active | % |