# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4436229 | 57; TUG-1907 | Stability | = | 100 | % | ALA4404889 | % | ||||
2. | ALA4436229 | 57; TUG-1907 | Stability | = | 100 | % | ALA4404888 | % | ||||
3. | ALA4436229 | 57; TUG-1907 | Activity | 0 | ALA4404886 | Not Active | ||||||
4. | ALA4436229 | 57; TUG-1907 | Activity | 0 | ALA4404885 | Active | Mus musculus | |||||
5. | ALA4436229 | 57; TUG-1907 | Stability | 0 | ALA4404884 | Unstable | % | |||||
6. | ALA4436229 | 57; TUG-1907 | Stability | = | 100 | % | ALA4404883 | % | ||||
7. | ALA4436229 | 57; TUG-1907 | INH | 0 | ALA4404882 | Not Active | % | Homo sapiens | ||||
8. | ALA4436229 | 57; TUG-1907 | Activity | 0 | ALA4404881 | Not Active | Homo sapiens | |||||
9. | ALA4436229 | 57; TUG-1907 | Activity | 0 | ALA4404880 | Not Active | Homo sapiens | |||||
10. | ALA4436229 | 57; TUG-1907 | Activity | 0 | ALA4404879 | Not Active | Homo sapiens | |||||
11. | ALA4436229 | 57; TUG-1907 | Activity | 0 | ALA4404878 | Not Active | Homo sapiens | |||||
12. | ALA4436229 | 57; TUG-1907 | F | = | 36 | % | ALA4404875 | % | ||||
13. | ALA4436229 | 57; TUG-1907 | AUC | = | 33800 | ng.min/ml | ALA4404874 | ng.hr.mL-1 | ||||
14. | ALA4436229 | 57; TUG-1907 | Cmax | = | 561 | ng/ml | ALA4404873 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
15. | ALA4436229 | 57; TUG-1907 | Tmax | = | 30 | min | ALA4404872 | hr | ||||
16. | ALA4436229 | 57; TUG-1907 | t1/2 | = | 63.5 | min | ALA4404871 | hr | ||||
17. | ALA4436229 | 57; TUG-1907 | CL | = | 70.3 | ml/min.kg | ALA4404870 | mL.min-1.kg-1 | ||||
18. | ALA4436229 | 57; TUG-1907 | Vd | = | 1150 | ml/kg | ALA4404869 | L.kg-1 | ||||
19. | ALA4436229 | 57; TUG-1907 | t1/2 | = | 11.4 | min | ALA4404868 | hr | ||||
20. | ALA4436229 | 57; TUG-1907 | Stability | = | 1 | % | ALA4404867 | % |