| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4437929 | 14 | Vdss | = | 9.8 | L/Kg | ALA4413831 | L.kg-1 | ||||
| 2. | ALA4437929 | 14 | beta t1/2 | = | 3.1 | hr | ALA4413830 | hr | ||||
| 3. | ALA4437929 | 14 | Tmax | = | 4 | hr | ALA4413829 | hr | ||||
| 4. | ALA4437929 | 14 | CL | = | 58 | ml/min.kg | ALA4413828 | mL.min-1.kg-1 | ||||
| 5. | ALA4437929 | 14 | Cmax | = | 0.16 | uM | ALA4413827 | nM | ||||
| 6. | ALA4437929 | 14 | F | = | 17.6 | % | ALA4413826 | % | ||||
| 7. | ALA4437929 | 14 | AUC | = | 1.41 | uM.hr | ALA4413825 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 8. | ALA4437929 | 14 | AUC | = | 0.64 | uM.hr | ALA4413824 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 9. | ALA4437929 | 14 | AUC | = | 1.02 | uM.hr | ALA4413823 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 10. | ALA4437929 | 14 | AUC | = | 0.58 | uM.hr | ALA4413822 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 11. | ALA4437929 | 14 | IC50 | > | 30 | uM | ALA4413821 | nM | Homo sapiens | |||
| 12. | ALA4437929 | 14 | Peff | = | 2.09 | 10'-6 cm/s | ALA4413820 | 10'-6 cm/s | ||||
| 13. | ALA4437929 | 14 | Stability | = | 19.7 | % | ALA4413819 | % | ||||
| 14. | ALA4437929 | 14 | Stability | = | 40 | % | ALA4413818 | % | ||||
| 15. | ALA4437929 | 14 | Stability | 0 | ALA4413817 | Not Determined | % | |||||
| 16. | ALA4437929 | 14 | Stability | = | 54.2 | % | ALA4413816 | % | ||||
| 17. | ALA4437929 | 14 | INH | = | 47 | % | ALA4413815 | % | Homo sapiens | |||
| 18. | ALA4437929 | 14 | INH | = | 31.1 | % | ALA4413814 | % | Homo sapiens | |||
| 19. | ALA4437929 | 14 | INH | = | 30.3 | % | ALA4413813 | % | Homo sapiens | |||
| 20. | ALA4437929 | 14 | INH | = | 26.6 | % | ALA4413812 | % | Homo sapiens |
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