# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4438120 | S-K1039 | IC50 | 0 | ALA4391937 | Not Determined | Homo sapiens | |||||
2. | ALA4438120 | S-K1039 | IC50 | = | 32 | uM | ALA4391939 | 4.50 | nM | Rattus norvegicus | ||
3. | ALA4438120 | S-K1039 | IC50 | = | 116 | uM | ALA4391936 | nM | Cricetulus griseus | |||
4. | ALA4438120 | S-K1039 | permeability | 0 | ALA4391932 | Impermeable | ||||||
5. | ALA4438120 | S-K1039 | INH | = | 46.4 | % | ALA4391930 | % | Homo sapiens | |||
6. | ALA4438120 | S-K1039 | Selectivity Index | = | 0.07 | ALA4391929 | Homo sapiens | |||||
7. | ALA4438120 | S-K1039 | IC50 | = | 40 | nM | ALA4391928 | 7.40 | nM | Homo sapiens | ||
8. | ALA4438120 | S-K1039 | IC50 | = | 580 | nM | ALA4391927 | 6.24 | nM | Homo sapiens |