Activities

JavaScript seems to be disabled in your browser. For the best experience on our site, be sure to turn on Javascript in your browser.

The page will load shortly, Thanks for your patience!

྾

Activities

Select ☑️ to add compounds to your custom library, then export your list as CSV / TSV. See how it works.

#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	ALA4438171	24; I-BET469	pIC50	=	7.9		ALA5218149	7.90		nM	Homo sapiens
2.	ALA4438171	24; I-BET469	pIC50	=	6.6		ALA5218148	6.60		nM	Homo sapiens
3.	ALA4438171	24; I-BET469	IC50	=	0.013	uM	ALA5127357	7.89		nM
4.	ALA4438171	24; I-BET469	pKd	=	8.3		ALA4404018	8.30		nM	Homo sapiens
5.	ALA4438171	24; I-BET469	Activity	=	65	%	ALA4404055			%	Mus musculus
6.	ALA4438171	24; I-BET469	Activity	=	65	%	ALA4404054			%	Mus musculus
7.	ALA4438171	24; I-BET469	Activity	=	20	%	ALA4404053			%	Mus musculus
8.	ALA4438171	24; I-BET469	Activity		0		ALA4404052		Active		Mus musculus
9.	ALA4438171	24; I-BET469	AUC	=	12503	ng.hr/ml	ALA4404051			ng.hr.mL-1
10.	ALA4438171	24; I-BET469	F	=	93	%	ALA4404050			%
11.	ALA4438171	24; I-BET469	AUC	=	26973	ng.hr/ml	ALA4404049			ng.hr.mL-1
12.	ALA4438171	24; I-BET469	AUC	=	2614	ng.hr/ml	ALA4404048			ng.hr.mL-1
13.	ALA4438171	24; I-BET469	AUC	=	3618	ng.hr/ml	ALA4404047			ng.hr.mL-1
14.	ALA4438171	24; I-BET469	Fu	=	7.2		ALA4404046
15.	ALA4438171	24; I-BET469	Stability	<	1	ml/min/g	ALA4404045			ml/min/g
16.	ALA4438171	24; I-BET469	Stability	<	0.48	ml/min/g	ALA4404044			ml/min/g
17.	ALA4438171	24; I-BET469	F	=	94	%	ALA4404043			%
18.	ALA4438171	24; I-BET469	Fu	=	0.72		ALA4404041
19.	ALA4438171	24; I-BET469	Stability	<	0.87	ml/min/g	ALA4404040			ml/min/g
20.	ALA4438171	24; I-BET469	Stability	<	0.4	ml/min/g	ALA4404039			ml/min/g