# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4438562 | 13 | permeability | = | 309 | nm/s | ALA4400129 | nm/s | ||||
2. | ALA4438562 | 13 | Ki | > | 15100 | nM | ALA4400128 | nM | Homo sapiens | |||
3. | ALA4438562 | 13 | Ki | > | 6150 | nM | ALA4400127 | nM | Homo sapiens | |||
4. | ALA4438562 | 13 | Ki | > | 15200 | nM | ALA4400126 | nM | Homo sapiens | |||
5. | ALA4438562 | 13 | Ki | > | 7160 | nM | ALA4400125 | nM | Homo sapiens | |||
6. | ALA4438562 | 13 | Ki | > | 6260 | nM | ALA4400124 | nM | Homo sapiens | |||
7. | ALA4438562 | 13 | Ki | > | 13300 | nM | ALA4400123 | nM | Homo sapiens | |||
8. | ALA4438562 | 13 | Ki | > | 3050 | nM | ALA4400122 | nM | Homo sapiens | |||
9. | ALA4438562 | 13 | Ki | > | 9000 | nM | ALA4400121 | nM | Homo sapiens | |||
10. | ALA4438562 | 13 | Ki | > | 27100 | nM | ALA4400120 | nM | Homo sapiens | |||
11. | ALA4438562 | 13 | Ki | = | 4850 | nM | ALA4400119 | 5.31 | nM | Homo sapiens | ||
12. | ALA4438562 | 13 | F | = | 15 | % | ALA4400117 | % | ||||
13. | ALA4438562 | 13 | t1/2 | = | 0.5 | hr | ALA4400113 | hr | ||||
14. | ALA4438562 | 13 | Vdss | = | 4.6 | L/Kg | ALA4400109 | L.kg-1 | ||||
15. | ALA4438562 | 13 | CL | = | 188 | ml/min.kg | ALA4400105 | mL.min-1.kg-1 | ||||
16. | ALA4438562 | 13 | AUC | = | 31 | nM.hr | ALA4400102 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
17. | ALA4438562 | 13 | permeability | = | 46 | nm/s | ALA4400101 | nm/s | ||||
18. | ALA4438562 | 13 | t1/2 | = | 6 | min | ALA4400099 | hr | ||||
19. | ALA4438562 | 13 | EC1.5 | = | 2.9 | uM | ALA4400098 | uM | Homo sapiens | |||
20. | ALA4438562 | 13 | Ki | = | 5.3 | nM | ALA4400097 | 8.28 | nM | Homo sapiens |