# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4440718 | 12 | Ratio | = | 4 | ALA4414886 | ||||||
2. | ALA4440718 | 12 | Ratio | = | 1 | ALA4414885 | ||||||
3. | ALA4440718 | 12 | Ratio | = | 0.5 | ALA4414884 | ||||||
4. | ALA4440718 | 12 | Ratio | = | 0.2 | ALA4414883 | ||||||
5. | ALA4440718 | 12 | Activity | 0 | ALA4414882 | Active | Mus musculus | |||||
6. | ALA4440718 | 12 | Activity | 0 | ALA4414881 | Active | Mus musculus | |||||
7. | ALA4440718 | 12 | Drug metabolism | 0 | ALA4414880 | Metabolite_Notdetected | ||||||
8. | ALA4440718 | 12 | INH | 0 | ALA4414879 | Dose-dependent effect | % | Mus musculus | ||||
9. | ALA4440718 | 12 | Drug uptake | = | 77 | nM | ALA4414850 | nM | ||||
10. | ALA4440718 | 12 | Drug uptake | = | 67 | nM | ALA4414849 | nM | ||||
11. | ALA4440718 | 12 | Drug uptake | = | 12 | nM | ALA4414848 | nM | ||||
12. | ALA4440718 | 12 | Drug uptake | = | 503 | nM | ALA4414843 | nM | ||||
13. | ALA4440718 | 12 | Drug uptake | = | 133 | nM | ALA4414842 | nM | ||||
14. | ALA4440718 | 12 | Drug uptake | = | 69 | nM | ALA4414841 | nM | ||||
15. | ALA4440718 | 12 | Drug uptake | = | 24 | nM | ALA4414840 | nM | ||||
16. | ALA4440718 | 12 | Ki(app) | = | 0 | uM | ALA4414854 | 10.15 | nM | Homo sapiens | ||
17. | ALA4440718 | 12 | Activity | 0 | ALA4414852 | Active | Mus musculus | |||||
18. | ALA4440718 | 12 | INH | 0 | ALA4414851 | Dose-dependent effect | % | Mus musculus | ||||
19. | ALA4440718 | 12 | INH | = | 91 | % | ALA4414847 | % | Mus musculus | |||
20. | ALA4440718 | 12 | INH | = | 77 | % | ALA4414846 | % | Mus musculus |