# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4441529 | 25 | pIC50 | = | 8.15 | ALA4394252 | 8.15 | nM | Mus musculus | |||
2. | ALA4441529 | 25 | INH | 0 | ALA4394262 | Active | % | |||||
3. | ALA4441529 | 25 | t1/2 | = | 1.3 | min | ALA4394260 | hr | ||||
4. | ALA4441529 | 25 | t1/2 | = | 0.64 | min | ALA4394259 | hr | ||||
5. | ALA4441529 | 25 | CLH | = | 2000 | ml/min.kg | ALA4394258 | mL.min-1.kg-1 | ||||
6. | ALA4441529 | 25 | CLH | = | 2700 | ml/min.kg | ALA4394250 | mL.min-1.kg-1 | ||||
7. | ALA4441529 | 25 | Ratio | = | 1.03 | ALA4394249 | ||||||
8. | ALA4441529 | 25 | Papp | = | 23 | 10'-6 cm/s | ALA4394248 | 10'-6 cm/s | ||||
9. | ALA4441529 | 25 | IC50 | > | 30 | uM | ALA4394243 | nM | Homo sapiens | |||
10. | ALA4441529 | 25 | INH | = | 7.1 | % | ALA4394251 | % | Homo sapiens | |||
11. | ALA4441529 | 25 | INH | = | 26 | % | ALA4394247 | % | Homo sapiens | |||
12. | ALA4441529 | 25 | INH | = | -4 | % | ALA4394246 | % | Homo sapiens | |||
13. | ALA4441529 | 25 | INH | = | 59 | % | ALA4394244 | % | Homo sapiens | |||
14. | ALA4441529 | 25 | INH | = | 72 | % | ALA4394245 | % | Homo sapiens | |||
15. | ALA4441529 | 25 | INH | 0 | ALA4394257 | Active | % | Homo sapiens | ||||
16. | ALA4441529 | 25 | INH | 0 | ALA4394256 | Active | % | Mus musculus | ||||
17. | ALA4441529 | 25 | Activity | 0 | ALA4394255 | Non-Toxic | Homo sapiens | |||||
18. | ALA4441529 | 25 | IC50 | = | 0.5 | nM | ALA4394254 | 9.30 | nM | |||
19. | ALA4441529 | 25 | IC50 | = | 7.1 | nM | ALA4394252 | 8.15 | nM | Mus musculus |