# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4441738 | 8a | AUC | = | 3.58 | microg.hr/mL | ALA4388750 | ng.hr.mL-1 | ||||
2. | ALA4441738 | 8a | Cmax | = | 1.54 | ug ml-1 | ALA4388749 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
3. | ALA4441738 | 8a | Activity | = | 88 | % | ALA4388737 | % | Homo sapiens | |||
4. | ALA4441738 | 8a | INH | = | 0 | % | ALA4388746 | % | Homo sapiens | |||
5. | ALA4441738 | 8a | INH | = | 3 | % | ALA4388745 | % | Homo sapiens | |||
6. | ALA4441738 | 8a | INH | = | 8 | % | ALA4388744 | % | Homo sapiens | |||
7. | ALA4441738 | 8a | INH | = | 7 | % | ALA4388743 | % | Homo sapiens | |||
8. | ALA4441738 | 8a | INH | = | 1 | % | ALA4388738 | % | Homo sapiens | |||
9. | ALA4441738 | 8a | Stability | = | 75 | % | ALA4388742 | % | ||||
10. | ALA4441738 | 8a | Stability | = | 93 | % | ALA4388741 | % | ||||
11. | ALA4441738 | 8a | solubility | = | 39 | ug ml-1 | ALA4388740 | ug.mL-1 | ||||
12. | ALA4441738 | 8a | EC200 | = | 0.025 | ug ml-1 | ALA4388739 | ug ml-1 | Mus musculus |