# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4442951 | DHD3; D2 | INH | 0 | ALA4378699 | Not Active | % | |||||
2. | ALA4442951 | DHD3; D2 | INH | 0 | ALA4378698 | Not Active | % | Homo sapiens | ||||
3. | ALA4442951 | DHD3; D2 | INH | 0 | ALA4378691 | Active | % | Homo sapiens | ||||
4. | ALA4442951 | DHD3; D2 | INH | 0 | ALA4378690 | Active | % | Homo sapiens | ||||
5. | ALA4442951 | DHD3; D2 | INH | 0 | ALA4378689 | Active | % | Homo sapiens | ||||
6. | ALA4442951 | DHD3; D2 | Activity | = | 84 | % | ALA4378688 | % | Homo sapiens | |||
7. | ALA4442951 | DHD3; D2 | Activity | = | 79 | % | ALA4378687 | % | Homo sapiens | |||
8. | ALA4442951 | DHD3; D2 | Activity | = | 45 | % | ALA4378686 | % | Homo sapiens | |||
9. | ALA4442951 | DHD3; D2 | CL | < | 2.9 | uL/min/pmol | ALA4378676 | uL/min/pmol | Homo sapiens | |||
10. | ALA4442951 | DHD3; D2 | CL | < | 5.8 | uL/min/pmol | ALA4378685 | uL/min/pmol | Homo sapiens | |||
11. | ALA4442951 | DHD3; D2 | CLH | = | 5 | microL/min/mg | ALA4378682 | mL.min-1.g-1 | ||||
12. | ALA4442951 | DHD3; D2 | CLH | < | 10 | microL/min/mg | ALA4378681 | mL.min-1.g-1 | ||||
13. | ALA4442951 | DHD3; D2 | CLH | = | 5 | microL/min/mg | ALA4378680 | mL.min-1.g-1 | ||||
14. | ALA4442951 | DHD3; D2 | CLH | = | 13 | microL/min/mg | ALA4378679 | mL.min-1.g-1 | ||||
15. | ALA4442951 | DHD3; D2 | t1/2 | = | 142 | min | ALA4378678 | hr | ||||
16. | ALA4442951 | DHD3; D2 | t1/2 | > | 138 | min | ALA4378677 | hr | ||||
17. | ALA4442951 | DHD3; D2 | t1/2 | = | 143 | min | ALA4378675 | hr | ||||
18. | ALA4442951 | DHD3; D2 | t1/2 | = | 112 | min | ALA4378674 | hr | ||||
19. | ALA4442951 | DHD3; D2 | PPB | = | 87.2 | % | ALA4378673 | % | ||||
20. | ALA4442951 | DHD3; D2 | PPB | = | 92.3 | % | ALA4378672 | % |