# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4444178 | 47 | IC50 | > | 30 | uM | ALA4414860 | nM | Homo sapiens | |||
2. | ALA4444178 | 47 | Ki(app) | = | 0.001 | uM | ALA4414854 | 9.10 | nM | Homo sapiens | ||
3. | ALA4444178 | 47 | AUClast | = | 6.61 | uM.hr | ALA4414839 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
4. | ALA4444178 | 47 | Cmax | = | 3.42 | uM | ALA4414838 | nM | ||||
5. | ALA4444178 | 47 | logP | = | 2.03 | ALA4414837 | ||||||
6. | ALA4444178 | 47 | t1/2 | = | 75 | min | ALA4414836 | hr | ||||
7. | ALA4444178 | 47 | t1/2 | = | 67 | min | ALA4414835 | hr | ||||
8. | ALA4444178 | 47 | t1/2 | = | 48 | min | ALA4414834 | hr | ||||
9. | ALA4444178 | 47 | t1/2 | = | 81 | min | ALA4414833 | hr | ||||
10. | ALA4444178 | 47 | t1/2 | = | 110 | min | ALA4414832 | hr | ||||
11. | ALA4444178 | 47 | IC50 | = | 0.34 | uM | ALA4414800 | 6.47 | nM | Mus musculus | ||
12. | ALA4444178 | 47 | Ratio | = | 7.7 | ALA4414796 | ||||||
13. | ALA4444178 | 47 | permeability | = | 69 | nm/s | ALA4414795 | nm/s | ||||
14. | ALA4444178 | 47 | IC50 | = | 0.23 | uM | ALA4414793 | 6.64 | nM | Homo sapiens | ||
15. | ALA4444178 | 47 | IC50 | = | 0.001 | uM | ALA4414790 | 8.89 | nM | Homo sapiens | ||
16. | ALA4444178 | 47 | IC50 | > | 50 | uM | ALA4414788 | nM | Homo sapiens | |||
17. | ALA4444178 | 47 | IC50 | > | 2 | uM | ALA4414787 | nM | Homo sapiens | |||
18. | ALA4444178 | 47 | IC50 | = | 50 | uM | ALA4414786 | 4.30 | nM | Homo sapiens | ||
19. | ALA4444178 | 47 | IC50 | = | 0.001 | uM | ALA4414785 | 8.89 | nM | Homo sapiens |