# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4445289 | (R)-18c | Time | > | 12 | hr | ALA4340589 | hr | Cavia porcellus | |||
2. | ALA4445289 | (R)-18c | Time | = | 1.9 | min | ALA4340588 | hr | Cavia porcellus | |||
3. | ALA4445289 | (R)-18c | Intrinsic activity | = | 0.97 | ALA4340587 | Cavia porcellus | |||||
4. | ALA4445289 | (R)-18c | pD2 | = | 7.02 | ALA4340586 | Cavia porcellus | |||||
5. | ALA4445289 | (R)-18c | Emax | = | 191.78 | % | ALA4340585 | % | Cavia porcellus | |||
6. | ALA4445289 | (R)-18c | Intrinsic activity | = | 84.79 | % | ALA4340584 | % | Homo sapiens | |||
7. | ALA4445289 | (R)-18c | Selectivity ratio | = | 5.68 | ALA4340583 | ||||||
8. | ALA4445289 | (R)-18c | pEC50 | = | 10.68 | ALA4340581 | 10.68 | nM | Homo sapiens | |||
9. | ALA4445289 | (R)-18c | EC50 | = | 21 | pM | ALA4340581 | 10.68 | nM | Homo sapiens | ||
10. | ALA4445289 | (R)-18c | pEC50 | = | 5 | ALA4340582 | 5.00 | nM | Homo sapiens |