# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Src Inhibitor 3 | 13 | Activity | 0 | ALA4308784 | Non-Toxic | ||||||
2. | Src Inhibitor 3 | 13 | Activity | 0 | ALA4308783 | Non-Toxic | ||||||
3. | Src Inhibitor 3 | 13 | FC | = | 2 | ALA4308780 | ||||||
4. | Src Inhibitor 3 | 13 | FC | = | 5.7 | ALA4308779 | ||||||
5. | Src Inhibitor 3 | 13 | t1/2 | = | 5.3 | hr | ALA4308778 | hr | ||||
6. | Src Inhibitor 3 | 13 | Ct | = | 1.3 | uM | ALA4308777 | uM | ||||
7. | Src Inhibitor 3 | 13 | Activity | 0 | ALA4308776 | Dose-dependent effect | ||||||
8. | Src Inhibitor 3 | 13 | Activity | 0 | ALA4308775 | Dose-dependent effect | ||||||
9. | Src Inhibitor 3 | 13 | Activity | = | -88 | % | ALA4308773 | % | Mus musculus | |||
10. | Src Inhibitor 3 | 13 | AUC | = | 221.5 | uM.hr | ALA4308771 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
11. | Src Inhibitor 3 | 13 | Tmax | = | 7 | hr | ALA4308770 | hr | ||||
12. | Src Inhibitor 3 | 13 | Cmax | = | 19.3 | uM | ALA4308769 | nM | ||||
13. | Src Inhibitor 3 | 13 | Fu | = | 0.3 | % | ALA4308768 | |||||
14. | Src Inhibitor 3 | 13 | Fu | < | 0.1 | % | ALA4308767 | |||||
15. | Src Inhibitor 3 | 13 | t1/2 | > | 120 | min | ALA4308766 | hr | ||||
16. | Src Inhibitor 3 | 13 | t1/2 | > | 120 | min | ALA4308765 | hr | ||||
17. | Src Inhibitor 3 | 13 | IC50 | = | 4 | nM | ALA4308764 | 8.40 | nM | Homo sapiens | ||
18. | Src Inhibitor 3 | 13 | Stability | = | 100 | % | ALA4308763 | % | ||||
19. | Src Inhibitor 3 | 13 | Stability | = | 91 | % | ALA4308762 | % | ||||
20. | Src Inhibitor 3 | 13 | Emax | = | 360 | % | ALA4308761 | % | Homo sapiens |