# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ML299 | 5; ML299 | IC50 | = | 6 | nM | ALA4329645 | 8.22 | nM | Homo sapiens | ||
2. | ML299 | 5; ML299 | IC50 | = | 20 | nM | ALA4329646 | 7.70 | nM | Homo sapiens | ||
3. | ML299 | 5; ML299 | CL free | > | 3800 | ml/min.kg | ALA5050792 | mL.min-1.kg-1 | ||||
4. | ML299 | 5; ML299 | CL | = | 36 | ml/min.kg | ALA5050791 | mL.min-1.kg-1 | ||||
5. | ML299 | 5; ML299 | Kinetic_solubility | = | 3.8 | ug ml-1 | ALA5050790 | ug.mL-1 | ||||
6. | ML299 | 5; ML299 | Ratio | = | 40 | ALA5050789 | ||||||
7. | ML299 | 5; ML299 | CLH | = | 312 | ml/min.kg | ALA5050788 | mL.min-1.kg-1 | ||||
8. | ML299 | 5; ML299 | CLH | = | 89 | ml/min.kg | ALA5050787 | mL.min-1.kg-1 | ||||
9. | ML299 | 5; ML299 | IC50 | = | 0.01 | uM | ALA5050786 | 8.00 | nM | Homo sapiens | ||
10. | ML299 | 5; ML299 | IC50 | = | 0.067 | uM | ALA5050785 | 7.17 | nM | Homo sapiens | ||
11. | ML299 | 5; ML299 | IC50 | = | 0.049 | uM | ALA5050784 | 7.31 | nM | Homo sapiens |