# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4446338 | THZ-P1-2 | Kd | = | 4.8 | nM | ALA4406349 | 8.32 | nM | Homo sapiens | ||
2. | ALA4446338 | THZ-P1-2 | Activity | = | 63 | % | ALA4406331 | % | Homo sapiens | |||
3. | ALA4446338 | THZ-P1-2 | Activity | = | 63 | % | ALA4406332 | % | Homo sapiens | |||
4. | ALA4446338 | THZ-P1-2 | IC50 | = | 40.1 | nM | ALA4345239 | 7.40 | nM | Homo sapiens | ||
5. | ALA4446338 | THZ-P1-2 | Activity | 0 | ALA4345238 | Active | Homo sapiens | |||||
6. | ALA4446338 | THZ-P1-2 | Activity | 0 | ALA4345237 | Active | Homo sapiens | |||||
7. | ALA4446338 | THZ-P1-2 | Activity | 0 | ALA4345236 | Active | Homo sapiens | |||||
8. | ALA4446338 | THZ-P1-2 | Activity | 0 | ALA4345235 | Active | Homo sapiens | |||||
9. | ALA4446338 | THZ-P1-2 | Activity | = | 6.4 | % | ALA4345234 | % | Homo sapiens | |||
10. | ALA4446338 | THZ-P1-2 | Activity | = | 4.3 | % | ALA4345233 | % | Homo sapiens | |||
11. | ALA4446338 | THZ-P1-2 | Activity | = | 1.3 | % | ALA4345232 | % | Homo sapiens | |||
12. | ALA4446338 | THZ-P1-2 | Activity | = | 0.9 | % | ALA4345231 | % | Homo sapiens | |||
13. | ALA4446338 | THZ-P1-2 | Activity | = | 0.1 | % | ALA4345230 | % | Homo sapiens | |||
14. | ALA4446338 | THZ-P1-2 | IC50 | = | 5.9 | uM | ALA4345229 | 5.23 | nM | Homo sapiens | ||
15. | ALA4446338 | THZ-P1-2 | IC50 | = | 0.95 | uM | ALA4345228 | 6.02 | nM | Homo sapiens | ||
16. | ALA4446338 | THZ-P1-2 | INH | = | 91 | % | ALA5045820 | % | Homo sapiens | |||
17. | ALA4446338 | THZ-P1-2 | IC50 | = | 950 | nM | ALA5260676 | 6.02 | nM | Homo sapiens |