| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4447951 | 24 | F | = | 83 | % | ALA4360348 | % | ||||
| 2. | ALA4447951 | 24 | Vdss | = | 2 | L/Kg | ALA4360347 | L.kg-1 | ||||
| 3. | ALA4447951 | 24 | CL | = | 54 | ml/min.Kg | ALA4360346 | mL.min-1.kg-1 | ||||
| 4. | ALA4447951 | 24 | CLH | = | 5 | uL/min | ALA4360342 | uL/min | ||||
| 5. | ALA4447951 | 24 | CL | < | 3 | uL/min.mg | ALA4360340 | mL.min-1.g-1 | ||||
| 6. | ALA4447951 | 24 | Fu | = | 10 | % | ALA4360341 | |||||
| 7. | ALA4447951 | 24 | logD | = | 2.06 | ALA4360338 | ||||||
| 8. | ALA4447951 | 24 | Therm_solubility | = | 94 | uM | ALA4360337 | nM | ||||
| 9. | ALA4447951 | 24 | GI50 | = | 0.46 | uM | ALA4360336 | nM | Homo sapiens | |||
| 10. | ALA4447951 | 24 | IC50 | = | 0.011 | uM | ALA4360335 | 7.96 | nM | |||
| 11. | ALA4447951 | 24 | IC50 | > | 40 | uM | ALA4360334 | nM | Homo sapiens | |||
| 12. | ALA4447951 | 24 | IC50 | = | 0.207 | uM | ALA4360333 | 6.68 | nM | Homo sapiens |
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