# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4449082 | 41g; RK-582 | GI50 | = | 230 | nM | ALA5227355 | nM | Homo sapiens | |||
2. | ALA4449082 | 41g; RK-582 | TGI | = | 71.1 | % | ALA5122247 | % | Homo sapiens | |||
3. | ALA4449082 | 41g; RK-582 | TGI | = | 68.8 | % | ALA5122246 | % | Homo sapiens | |||
4. | ALA4449082 | 41g; RK-582 | TGI | = | 52 | % | ALA5122245 | % | Homo sapiens | |||
5. | ALA4449082 | 41g; RK-582 | F | = | 100 | % | ALA5122244 | % | ||||
6. | ALA4449082 | 41g; RK-582 | IC50 | = | 1.24 | uM | ALA5122239 | 5.91 | nM | Homo sapiens | ||
7. | ALA4449082 | 41g; RK-582 | IC50 | = | 18.187 | uM | ALA5122238 | 4.74 | nM | Homo sapiens | ||
8. | ALA4449082 | 41g; RK-582 | IC50 | = | 0.039 | uM | ALA5122237 | 7.41 | nM | Homo sapiens | ||
9. | ALA4449082 | 41g; RK-582 | IC50 | = | 0.036 | uM | ALA5122236 | 7.44 | nM | Homo sapiens | ||
10. | ALA4449082 | 41g; RK-582 | TGI | = | 52.3 | % | ALA5122235 | % | Homo sapiens | |||
11. | ALA4449082 | 41g; RK-582 | FC | = | 0.39 | ALA4345481 | Homo sapiens | |||||
12. | ALA4449082 | 41g; RK-582 | Activity | 0 | ALA4345477 | Toxic | ||||||
13. | ALA4449082 | 41g; RK-582 | Activity | 0 | ALA4345476 | Toxic | ||||||
14. | ALA4449082 | 41g; RK-582 | Activity | 0 | ALA4345475 | Toxic | ||||||
15. | ALA4449082 | 41g; RK-582 | Activity | 0 | ALA4345474 | Toxic | ||||||
16. | ALA4449082 | 41g; RK-582 | Activity | 0 | ALA4345473 | Toxic | ||||||
17. | ALA4449082 | 41g; RK-582 | Cp | = | 26.9 | umol/L | ALA4345472 | umol/L | ||||
18. | ALA4449082 | 41g; RK-582 | Cp | = | 23.3 | umol/L | ALA4345471 | umol/L | ||||
19. | ALA4449082 | 41g; RK-582 | Cp | = | 10.1 | umol/L | ALA4345470 | umol/L | ||||
20. | ALA4449082 | 41g; RK-582 | INH | 0 | ALA4345469 | Active | % | Mus musculus |