| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4449557 | 10; NTRC 0066-0 | IC50 | = | 0.6 | nM | ALA5227240 | 9.22 | nM | Homo sapiens | ||
| 2. | ALA4449557 | 10; NTRC 0066-0 | t1/2 | = | 2.9 | hr | ALA4349534 | hr | ||||
| 3. | ALA4449557 | 10; NTRC 0066-0 | Cmax | = | 3060 | nmol/L | ALA4349535 | nM | ||||
| 4. | ALA4449557 | 10; NTRC 0066-0 | t1/2 | = | 3.4 | hr | ALA4349532 | hr | ||||
| 5. | ALA4449557 | 10; NTRC 0066-0 | Cmax | = | 629 | nmol/L | ALA4349533 | nM | ||||
| 6. | ALA4449557 | 10; NTRC 0066-0 | t1/2 | = | 3.9 | hr | ALA4349553 | hr | ||||
| 7. | ALA4449557 | 10; NTRC 0066-0 | Cmax | = | 188 | nmol/L | ALA4349554 | nM | ||||
| 8. | ALA4449557 | 10; NTRC 0066-0 | F | = | 45.2 | % | ALA4349555 | % | ||||
| 9. | ALA4449557 | 10; NTRC 0066-0 | F | = | 90.3 | % | ALA4349556 | % | ||||
| 10. | ALA4449557 | 10; NTRC 0066-0 | IC50 | < | 1 | nM | ALA5042273 | nM | Homo sapiens | |||
| 11. | ALA4449557 | 10; NTRC 0066-0 | deltaTm | = | 21.6 | degrees C | ALA5042246 | degrees C | Homo sapiens | |||
| 12. | ALA4449557 | 10; NTRC 0066-0 | IC50 | = | 4.7 | nM | ALA5042245 | 8.33 | nM | Homo sapiens | ||
| 13. | ALA4449557 | 10; NTRC 0066-0 | deltaTm | = | 13.2 | degrees C | ALA5042235 | degrees C | Homo sapiens | |||
| 14. | ALA4449557 | 10; NTRC 0066-0 | IC50 | = | 0.9 | nM | ALA5037592 | 9.05 | nM | Homo sapiens |
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