# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4451030 | 48; UR-AP148 | Ratio Ki | = | 400 | ALA4397801 | Homo sapiens | |||||
2. | ALA4451030 | 48; UR-AP148 | Ratio Ki | = | 60 | ALA4397800 | Homo sapiens | |||||
3. | ALA4451030 | 48; UR-AP148 | Ratio Ki | = | 6500 | ALA4397799 | Homo sapiens | |||||
4. | ALA4451030 | 48; UR-AP148 | Ratio Ki | = | 49 | ALA4397798 | Homo sapiens | |||||
5. | ALA4451030 | 48; UR-AP148 | pKi | = | 6.37 | ALA4397797 | 6.37 | nM | Homo sapiens | |||
6. | ALA4451030 | 48; UR-AP148 | pKi | = | 7.21 | ALA4397796 | 7.21 | nM | Homo sapiens | |||
7. | ALA4451030 | 48; UR-AP148 | pKi | = | 5.17 | ALA4397795 | 5.17 | nM | Homo sapiens | |||
8. | ALA4451030 | 48; UR-AP148 | pKi | = | 8.97 | ALA4397794 | 8.97 | nM | Homo sapiens | |||
9. | ALA4451030 | 48; UR-AP148 | pKi | = | 7.38 | ALA4397793 | 7.38 | nM | Homo sapiens | |||
10. | ALA4451030 | 48; UR-AP148 | pIC50 | = | 7.38 | ALA4397809 | 7.38 | nM | Homo sapiens | |||
11. | ALA4451030 | 48; UR-AP148 | pIC50 | = | 8.48 | ALA4397808 | 8.48 | nM | Homo sapiens | |||
12. | ALA4451030 | 48; UR-AP148 | pIC50 | = | 7.03 | ALA4397803 | 7.03 | nM | Homo sapiens | |||
13. | ALA4451030 | 48; UR-AP148 | Activity | > | 95 | % | ALA4397810 | % | Homo sapiens | |||
14. | ALA4451030 | 48; UR-AP148 | pKi | = | 8.69 | ALA4397809 | 8.69 | nM | Homo sapiens | |||
15. | ALA4451030 | 48; UR-AP148 | pKi | = | 8.97 | ALA4397808 | 8.97 | nM | Homo sapiens | |||
16. | ALA4451030 | 48; UR-AP148 | Stability | > | 99 | % | ALA4397807 | % | ||||
17. | ALA4451030 | 48; UR-AP148 | Stability | > | 99 | % | ALA4397806 | % | ||||
18. | ALA4451030 | 48; UR-AP148 | Stability | > | 99 | % | ALA4397805 | % | ||||
19. | ALA4451030 | 48; UR-AP148 | Stability | = | 99 | % | ALA4397804 | % | ||||
20. | ALA4451030 | 48; UR-AP148 | INH | 0 | ALA4397803 | Dose-dependent effect | % | Homo sapiens |