# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4451878 | 26, Diastereomer A | Ratio IC50 | = | 4.5 | ALA4407252 | Homo sapiens | |||||
2. | ALA4451878 | 26, Diastereomer A | INH | 0 | ALA4407251 | Dose-dependent effect | % | Homo sapiens | ||||
3. | ALA4451878 | 26, Diastereomer A | Activity | = | 5 | % | ALA4407245 | % | Homo sapiens | |||
4. | ALA4451878 | 26, Diastereomer A | Activity | = | 6 | % | ALA4407244 | % | Homo sapiens | |||
5. | ALA4451878 | 26, Diastereomer A | Activity | = | 8 | % | ALA4407243 | % | Homo sapiens | |||
6. | ALA4451878 | 26, Diastereomer A | INH | = | 44 | % | ALA4407241 | % | Homo sapiens | |||
7. | ALA4451878 | 26, Diastereomer A | INH | = | 32 | % | ALA4407240 | % | Homo sapiens | |||
8. | ALA4451878 | 26, Diastereomer A | INH | = | -3 | % | ALA4407239 | % | Homo sapiens | |||
9. | ALA4451878 | 26, Diastereomer A | Cp | = | 48.7 | ng/ml | ALA4407238 | ng/ml | ||||
10. | ALA4451878 | 26, Diastereomer A | IC50 | = | 0.06 | uM | ALA4407236 | 7.22 | nM | Rattus norvegicus | ||
11. | ALA4451878 | 26, Diastereomer A | Activity | = | 81.9 | % | ALA4407235 | % | Homo sapiens | |||
12. | ALA4451878 | 26, Diastereomer A | Activity | = | 94.9 | % | ALA4407234 | % | Homo sapiens | |||
13. | ALA4451878 | 26, Diastereomer A | Activity | = | 115 | % | ALA4407233 | % | Homo sapiens | |||
14. | ALA4451878 | 26, Diastereomer A | IC50 | = | 0.02 | uM | ALA4407232 | 7.70 | nM | Homo sapiens | ||
15. | ALA4451878 | 26, Diastereomer A | IC50 | = | 0.14 | uM | ALA4407232 | 6.85 | nM | Homo sapiens | ||
16. | ALA4451878 | 26, Diastereomer A | INH | = | 100 | % | ALA4407231 | % | Homo sapiens | |||
17. | ALA4451878 | 26, Diastereomer A | INH | = | 98 | % | ALA4407231 | % | Homo sapiens | |||
18. | ALA4451878 | 26, Diastereomer A | INH | = | 98 | % | ALA4407230 | % | Homo sapiens | |||
19. | ALA4451878 | 26, Diastereomer A | INH | = | 95 | % | ALA4407230 | % | Homo sapiens | |||
20. | ALA4451878 | 26, Diastereomer A | INH | = | 84 | % | ALA4407229 | % | Homo sapiens |