# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4452527 | 14; SD-36 | Activity | > | 50 | % | ALA5242542 | % | Homo sapiens | |||
2. | ALA4452527 | 14; SD-36 | Activity | > | 50 | % | ALA5242541 | % | Homo sapiens | |||
3. | ALA4452527 | 14; SD-36 | Activity | > | 50 | % | ALA5242540 | % | Homo sapiens | |||
4. | ALA4452527 | 14; SD-36 | Activity | > | 90 | % | ALA5242539 | % | Homo sapiens | |||
5. | ALA4452527 | 14; SD-36 | Kd | = | 1 | uM | ALA5124525 | 6.00 | nM | Homo sapiens | ||
6. | ALA4452527 | 14; SD-36 | Kd | = | 1 | uM | ALA5124524 | 6.00 | nM | Homo sapiens | ||
7. | ALA4452527 | 14; SD-36 | Kd | = | 44 | nM | ALA5124523 | 7.36 | nM | Homo sapiens | ||
8. | ALA4452527 | 14; SD-36 | Drug metabolism | = | 10 | % | ALA4715529 | % | ||||
9. | ALA4452527 | 14; SD-36 | Drug metabolism | 0 | ALA4715526 | Metabolite_Notdetected | ||||||
10. | ALA4452527 | 14; SD-36 | Drug metabolism | 0 | ALA4715525 | Metabolite_Detected | ||||||
11. | ALA4452527 | 14; SD-36 | Drug metabolism | = | 50 | % | ALA4715524 | % | ||||
12. | ALA4452527 | 14; SD-36 | Drug metabolism | = | 25 | % | ALA4715523 | % | ||||
13. | ALA4452527 | 14; SD-36 | t1/2 | = | 4 | hr | ALA4715522 | hr | ||||
14. | ALA4452527 | 14; SD-36 | t1/2 | = | 22 | hr | ALA4715521 | hr | ||||
15. | ALA4452527 | 14; SD-36 | Drug metabolism | = | 4 | % | ALA4715520 | % | ||||
16. | ALA4452527 | 14; SD-36 | Drug metabolism | 0 | ALA4715519 | Metabolite_Notdetected | ||||||
17. | ALA4452527 | 14; SD-36 | Drug metabolism | = | 90 | % | ALA4715518 | % | ||||
18. | ALA4452527 | 14; SD-36 | Drug metabolism | = | 50 | % | ALA4715517 | % | ||||
19. | ALA4452527 | 14; SD-36 | Drug uptake | = | 396 | ng/g | ALA4715513 | ng/g | ||||
20. | ALA4452527 | 14; SD-36 | Drug uptake | = | 1750 | ng/g | ALA4715512 | ng/g |