| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4456515 | 12 | F | = | 48.6 | % | ALA4355768 | % | ||||
| 2. | ALA4456515 | 12 | Vdss | = | 1.33 | L/Kg | ALA4355765 | L.kg-1 | ||||
| 3. | ALA4456515 | 12 | t1/2 | = | 1.29 | hr | ALA4355762 | hr | ||||
| 4. | ALA4456515 | 12 | CL | = | 33.6 | ml/min.kg | ALA4355760 | mL.min-1.kg-1 | ||||
| 5. | ALA4456515 | 12 | AUC/dose | = | 0.903 | uM.hr.kg/mg | ALA4355759 | uM.hr.kg/mg | ||||
| 6. | ALA4456515 | 12 | Ki | > | 10000 | nM | ALA4355756 | nM | Homo sapiens | |||
| 7. | ALA4456515 | 12 | EC50 | = | 509 | nM | ALA4355755 | 6.29 | nM | Rattus norvegicus | ||
| 8. | ALA4456515 | 12 | Ki | = | 5.6 | nM | ALA4355754 | 8.25 | nM | Homo sapiens | ||
| 9. | ALA4456515 | 12 | Papp | = | 2.2 | 10'-6 cm/s | ALA4355751 | 10'-6 cm/s |
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