| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4457100 | 10 | logD | = | 1.7 | ALA4400307 | ||||||
| 2. | ALA4457100 | 10 | logP | = | 4.2 | ALA4400306 | ||||||
| 3. | ALA4457100 | 10 | Kinetic_solubility | = | 250 | uM | ALA4400305 | nM | ||||
| 4. | ALA4457100 | 10 | solubility | > | 50 | mM | ALA4400304 | nM | ||||
| 5. | ALA4457100 | 10 | Activity | = | 52.3 | % | ALA4400303 | % | Rattus norvegicus | |||
| 6. | ALA4457100 | 10 | Ratio | = | 3.02 | ALA4400302 | ||||||
| 7. | ALA4457100 | 10 | Ratio | = | 0.24 | ALA4400301 | ||||||
| 8. | ALA4457100 | 10 | Tmax | = | 1 | hr | ALA4400300 | hr | ||||
| 9. | ALA4457100 | 10 | F | = | 62.3 | % | ALA4400299 | % | ||||
| 10. | ALA4457100 | 10 | Fm | = | 99 | % | ALA4400298 | % | ||||
| 11. | ALA4457100 | 10 | Fm | = | 99 | % | ALA4400297 | % | ||||
| 12. | ALA4457100 | 10 | ED50 | = | 0.47 | mg kg-1 | ALA4400296 | mg.kg-1 | Rattus norvegicus | |||
| 13. | ALA4457100 | 10 | IC50 | = | 17.5 | uM | ALA4400294 | 4.76 | nM | Homo sapiens | ||
| 14. | ALA4457100 | 10 | Ki | = | 4700 | nM | ALA4400291 | 5.33 | nM | Rattus norvegicus | ||
| 15. | ALA4457100 | 10 | Ki | = | 9 | nM | ALA4400290 | 8.05 | nM | Rattus norvegicus | ||
| 16. | ALA4457100 | 10 | Ki | = | 3 | nM | ALA4400289 | 8.52 | nM | Homo sapiens |
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