# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4457171 | (-)-8a, D-593 | Ratio EC50 | = | 8.74 | ALA4430345 | ||||||
2. | ALA4457171 | (-)-8a, D-593 | INH | 0 | ALA4430343 | Active | % | Homo sapiens | ||||
3. | ALA4457171 | (-)-8a, D-593 | Activity | = | 18 | % | ALA4430342 | % | Rattus norvegicus | |||
4. | ALA4457171 | (-)-8a, D-593 | Activity | 0 | ALA4430341 | Dose-dependent effect | Rattus norvegicus | |||||
5. | ALA4457171 | (-)-8a, D-593 | Activity | 0 | ALA4430340 | Active | Rattus norvegicus | |||||
6. | ALA4457171 | (-)-8a, D-593 | Emax | = | 83.4 | % | ALA4430339 | % | Homo sapiens | |||
7. | ALA4457171 | (-)-8a, D-593 | EC50 | = | 2.62 | nM | ALA4430338 | 8.58 | nM | Homo sapiens | ||
8. | ALA4457171 | (-)-8a, D-593 | Emax | = | 97.4 | % | ALA4430337 | % | Homo sapiens | |||
9. | ALA4457171 | (-)-8a, D-593 | EC50 | = | 22.9 | nM | ALA4430336 | 7.64 | nM | Homo sapiens | ||
10. | ALA4457171 | (-)-8a, D-593 | Ratio Ki | = | 46 | ALA4430335 | ||||||
11. | ALA4457171 | (-)-8a, D-593 | Ki | = | 1.42 | nM | ALA4430334 | 8.85 | nM | Rattus norvegicus | ||
12. | ALA4457171 | (-)-8a, D-593 | Ki | = | 65.7 | nM | ALA4430333 | 7.18 | nM | Rattus norvegicus |