# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4457578 | 12k; PXS-5120A | INH | 0 | ALA4323333 | Active | % | Homo sapiens | ||||
2. | ALA4457578 | 12k; PXS-5120A | F | < | 1 | % | ALA4323307 | % | ||||
3. | ALA4457578 | 12k; PXS-5120A | F | < | 1 | % | ALA4323306 | % | ||||
4. | ALA4457578 | 12k; PXS-5120A | Kinact | = | 0.89 | /min | ALA4323325 | /min | Homo sapiens | |||
5. | ALA4457578 | 12k; PXS-5120A | IC50 | = | 13 | nM | ALA4323323 | 7.89 | nM | Homo sapiens | ||
6. | ALA4457578 | 12k; PXS-5120A | FC | = | 1 | ALA4323305 | Homo sapiens | |||||
7. | ALA4457578 | 12k; PXS-5120A | Imax | > | 80 | % | ALA4323303 | % | Homo sapiens | |||
8. | ALA4457578 | 12k; PXS-5120A | INH | 0 | ALA4323302 | Active | % | Homo sapiens | ||||
9. | ALA4457578 | 12k; PXS-5120A | Ki | = | 83 | nM | ALA4323301 | 7.08 | nM | Homo sapiens | ||
10. | ALA4457578 | 12k; PXS-5120A | t1/2 | > | 120 | min | ALA4323300 | hr | ||||
11. | ALA4457578 | 12k; PXS-5120A | t1/2 | > | 120 | min | ALA4323299 | hr | ||||
12. | ALA4457578 | 12k; PXS-5120A | t1/2 | > | 120 | min | ALA4323298 | hr | ||||
13. | ALA4457578 | 12k; PXS-5120A | t1/2 | > | 90 | min | ALA4323297 | hr | ||||
14. | ALA4457578 | 12k; PXS-5120A | t1/2 | > | 90 | min | ALA4323296 | hr | ||||
15. | ALA4457578 | 12k; PXS-5120A | t1/2 | > | 90 | min | ALA4323295 | hr | ||||
16. | ALA4457578 | 12k; PXS-5120A | t1/2 | > | 120 | min | ALA4323294 | hr | ||||
17. | ALA4457578 | 12k; PXS-5120A | t1/2 | > | 120 | min | ALA4323293 | hr | ||||
18. | ALA4457578 | 12k; PXS-5120A | t1/2 | > | 120 | min | ALA4323292 | hr | ||||
19. | ALA4457578 | 12k; PXS-5120A | PPB | = | 92 | % | ALA4323291 | % | ||||
20. | ALA4457578 | 12k; PXS-5120A | PPB | = | 86 | % | ALA4323290 | % |