# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4457739 | 19 | Drug metabolism | < | 100 | pmol/mg.hr | ALA4325062 | pmol/mg.hr | ||||
2. | ALA4457739 | 19 | CLH | > | 1250 | uL/min.mg | ALA4325035 | mL.min-1.g-1 | ||||
3. | ALA4457739 | 19 | CLH | = | 15.4 | uL/min | ALA4325034 | uL/min | ||||
4. | ALA4457739 | 19 | solubility | 0 | ALA4325080 | Insoluble | ||||||
5. | ALA4457739 | 19 | solubility | = | 25 | mg/ml | ALA4325077 | ug.mL-1 | ||||
6. | ALA4457739 | 19 | Ratio | = | 4 | ALA4325070 | ||||||
7. | ALA4457739 | 19 | Activity | 0 | ALA4325069 | Not Active | ||||||
8. | ALA4457739 | 19 | fAUC | = | 291 | ng.hr/ml | ALA4325068 | ng.hr.mL-1 | ||||
9. | ALA4457739 | 19 | Activity | 0 | ALA4325066 | Not Determined | Homo sapiens | |||||
10. | ALA4457739 | 19 | IC50 | > | 50 | uM | ALA4325065 | nM | Homo sapiens | |||
11. | ALA4457739 | 19 | IC50 | > | 50 | uM | ALA4325064 | nM | Homo sapiens | |||
12. | ALA4457739 | 19 | IC50 | > | 50 | uM | ALA4325063 | nM | Homo sapiens | |||
13. | ALA4457739 | 19 | MIC90 | > | 16 | ug ml-1 | ALA4325061 | ug.mL-1 | Stenotrophomonas maltophilia | |||
14. | ALA4457739 | 19 | MIC90 | = | 1 | ug ml-1 | ALA4325060 | ug.mL-1 | Pseudomonas aeruginosa | |||
15. | ALA4457739 | 19 | MIC90 | > | 16 | ug ml-1 | ALA4325059 | ug.mL-1 | Moraxella catarrhalis | |||
16. | ALA4457739 | 19 | MIC90 | <= | 0.03 | ug ml-1 | ALA4325058 | ug.mL-1 | Haemophilus influenzae | |||
17. | ALA4457739 | 19 | MIC90 | = | 4 | ug ml-1 | ALA4325057 | ug.mL-1 | Burkholderia cepacia | |||
18. | ALA4457739 | 19 | MIC90 | > | 16 | ug ml-1 | ALA4325056 | ug.mL-1 | Acinetobacter baumannii | |||
19. | ALA4457739 | 19 | MIC90 | = | 0.25 | ug ml-1 | ALA4325055 | ug.mL-1 | Serratia marcescens | |||
20. | ALA4457739 | 19 | MIC90 | = | 0.5 | ug ml-1 | ALA4325054 | ug.mL-1 | Proteus mirabilis |