# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4459416 | S-K1040 | IC50 | 0 | ALA4391937 | Not Determined | Homo sapiens | |||||
2. | ALA4459416 | S-K1040 | IC50 | = | 18 | uM | ALA4391939 | 4.75 | nM | Rattus norvegicus | ||
3. | ALA4459416 | S-K1040 | IC50 | = | 34 | uM | ALA4391936 | 4.47 | nM | Cricetulus griseus | ||
4. | ALA4459416 | S-K1040 | permeability | 0 | ALA4391932 | Permeable | ||||||
5. | ALA4459416 | S-K1040 | INH | = | 59.1 | % | ALA4391930 | % | Homo sapiens | |||
6. | ALA4459416 | S-K1040 | Selectivity Index | = | 0.1 | ALA4391929 | Homo sapiens | |||||
7. | ALA4459416 | S-K1040 | IC50 | = | 123 | nM | ALA4391928 | 6.91 | nM | Homo sapiens | ||
8. | ALA4459416 | S-K1040 | IC50 | = | 1300 | nM | ALA4391927 | 5.89 | nM | Homo sapiens |