# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4459585 | 10; PF-06826647 | IC50 | = | 17 | nM | ALA4377467 | 7.77 | nM | Homo sapiens | ||
2. | ALA4459585 | 10; PF-06826647 | IC50 | > | 10000 | nM | ALA4377466 | nM | Homo sapiens | |||
3. | ALA4459585 | 10; PF-06826647 | IC50 | = | 74 | nM | ALA4377465 | 7.13 | nM | Homo sapiens | ||
4. | ALA4459585 | 10; PF-06826647 | IC50 | = | 383 | nM | ALA4377464 | 6.42 | nM | Homo sapiens | ||
5. | ALA4459585 | 10; PF-06826647 | Activity | = | 31.3 | % | ALA4675864 | % | Mus musculus | |||
6. | ALA4459585 | 10; PF-06826647 | Activity | = | 34 | % | ALA4675863 | % | Mus musculus | |||
7. | ALA4459585 | 10; PF-06826647 | Activity | = | 46.2 | % | ALA4675862 | % | Mus musculus | |||
8. | ALA4459585 | 10; PF-06826647 | Activity | 0 | ALA4675861 | Not Active | Mus musculus | |||||
9. | ALA4459585 | 10; PF-06826647 | Activity | = | 98 | % | ALA4675860 | % | Mus musculus | |||
10. | ALA4459585 | 10; PF-06826647 | Activity | = | 94 | % | ALA4675859 | % | Mus musculus | |||
11. | ALA4459585 | 10; PF-06826647 | Activity | = | 77 | % | ALA4675858 | % | Mus musculus | |||
12. | ALA4459585 | 10; PF-06826647 | Activity | = | 51 | % | ALA4675857 | % | Mus musculus | |||
13. | ALA4459585 | 10; PF-06826647 | Drug uptake(free) | = | 668 | nM | ALA4675856 | nM | ||||
14. | ALA4459585 | 10; PF-06826647 | Drug uptake(free) | = | 225 | nM | ALA4675855 | nM | ||||
15. | ALA4459585 | 10; PF-06826647 | Drug uptake(free) | = | 45.7 | nM | ALA4675854 | nM | ||||
16. | ALA4459585 | 10; PF-06826647 | Drug uptake(free) | = | 14.5 | nM | ALA4675853 | nM | ||||
17. | ALA4459585 | 10; PF-06826647 | IC50 | = | 2220 | nM | ALA4675852 | 5.65 | nM | Homo sapiens | ||
18. | ALA4459585 | 10; PF-06826647 | IC50 | = | 3740 | nM | ALA4675851 | 5.43 | nM | Homo sapiens | ||
19. | ALA4459585 | 10; PF-06826647 | IC50 | = | 4840 | nM | ALA4675850 | 5.32 | nM | Homo sapiens | ||
20. | ALA4459585 | 10; PF-06826647 | IC50 | = | 4890 | nM | ALA4675849 | 5.31 | nM | Homo sapiens |