# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4459996 | 25 | Kinetic_solubility | = | 1.4 | 10'-5mg/ml | ALA4384339 | 10'-5mg/ml | ||||
2. | ALA4459996 | 25 | Kinetic_solubility | = | 1.7 | 10'-5mg/ml | ALA4384338 | 10'-5mg/ml | ||||
3. | ALA4459996 | 25 | CLH | < | 3 | ml/min | ALA4384337 | ml/min | ||||
4. | ALA4459996 | 25 | t1/2 | > | 231 | min | ALA4384336 | hr | ||||
5. | ALA4459996 | 25 | EC50 | = | 0.7 | uM | ALA4384334 | 6.16 | nM | Mus musculus | ||
6. | ALA4459996 | 25 | Activity | = | 11000 | % | ALA4384331 | % | Mus musculus | |||
7. | ALA4459996 | 25 | IC50 | = | 0.6 | uM | ALA4384330 | 6.22 | nM | |||
8. | ALA4459996 | 25 | Activity | = | 89 | % | ALA4384328 | % | Mus musculus | |||
9. | ALA4459996 | 25 | IC50 | = | 2.3 | uM | ALA4384327 | 5.64 | nM | |||
10. | ALA4459996 | 25 | INH | = | 3.3 | % | ALA4384324 | % |