# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4464968 | 17; APY-d3 | IC50 | = | 17 | nM | ALA4433135 | 7.77 | nM | Homo sapiens | ||
2. | ALA4464968 | 17; APY-d3 | IC50 | = | 20 | nM | ALA4433140 | 7.70 | nM | Mus musculus | ||
3. | ALA4464968 | 17; APY-d3 | INH | 0 | ALA4433155 | Active | % | Homo sapiens | ||||
4. | ALA4464968 | 17; APY-d3 | Activity | 0 | ALA4433153 | Non-Toxic | Mus musculus | |||||
5. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433152 | ||||||
6. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433151 | ||||||
7. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433150 | ||||||
8. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433149 | ||||||
9. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433148 | ||||||
10. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433147 | ||||||
11. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433146 | ||||||
12. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433145 | ||||||
13. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433144 | ||||||
14. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433143 | ||||||
15. | ALA4464968 | 17; APY-d3 | Ratio IC50 | > | 100 | ALA4433142 | ||||||
16. | ALA4464968 | 17; APY-d3 | Stability | 0 | ALA4433141 | Stable | % | |||||
17. | ALA4464968 | 17; APY-d3 | INH | 0 | ALA4433139 | Active | % | |||||
18. | ALA4464968 | 17; APY-d3 | IC50 | = | 0.24 | uM | ALA4433138 | 6.62 | nM | Homo sapiens | ||
19. | ALA4464968 | 17; APY-d3 | Kd | = | 27 | nM | ALA4433137 | 7.57 | nM | Homo sapiens | ||
20. | ALA4464968 | 17; APY-d3 | t1/2 | > | 72 | hr | ALA4433136 | hr |