| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4468523 | 38 | Activity | 0 | ALA4397526 | Not Active | Rattus norvegicus | |||||
| 2. | ALA4468523 | 38 | Activity | 0 | ALA4397525 | Not Active | Rattus norvegicus | |||||
| 3. | ALA4468523 | 38 | t1/2 | = | 20 | min | ALA4397523 | hr | ||||
| 4. | ALA4468523 | 38 | Activity | = | 80 | % | ALA4397521 | % | Rattus norvegicus | |||
| 5. | ALA4468523 | 38 | Ratio EC50 | = | 10 | ALA4397520 | ||||||
| 6. | ALA4468523 | 38 | Activity | = | 1.3 | g | ALA4397519 | g | Rattus norvegicus | |||
| 7. | ALA4468523 | 38 | Activity | = | 5 | g | ALA4397517 | g | Rattus norvegicus | |||
| 8. | ALA4468523 | 38 | EC50 | = | 0.64 | pM | ALA4397516 | nM | Rattus norvegicus | |||
| 9. | ALA4468523 | 38 | Activity | 0 | ALA4397515 | Dose-dependent effect | Rattus norvegicus | |||||
| 10. | ALA4468523 | 38 | beta t1/2 | = | 16 | min | ALA4397514 | hr | ||||
| 11. | ALA4468523 | 38 | Efficacy | = | 99 | % | ALA4397513 | % | Rattus norvegicus | |||
| 12. | ALA4468523 | 38 | EC50 | = | 0.02 | nM | ALA4397512 | 10.70 | nM | Rattus norvegicus | ||
| 13. | ALA4468523 | 38 | Activity | 0 | ALA4397511 | Not Active | Homo sapiens | |||||
| 14. | ALA4468523 | 38 | PPB | = | 85 | % | ALA4397510 | % | ||||
| 15. | ALA4468523 | 38 | CL | = | 57 | % | ALA4397509 | % | ||||
| 16. | ALA4468523 | 38 | CL | = | 14 | ml/min.Kg | ALA4397508 | mL.min-1.kg-1 | ||||
| 17. | ALA4468523 | 38 | Activity | 0 | ALA4397507 | Not Active | Homo sapiens | |||||
| 18. | ALA4468523 | 38 | Ratio EC50 | = | 1500 | ALA4397506 | ||||||
| 19. | ALA4468523 | 38 | EC50 | = | 110 | nM | ALA4397503 | 6.96 | nM | Homo sapiens | ||
| 20. | ALA4468523 | 38 | EC50 | = | 0.07 | nM | ALA4397500 | 10.15 | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!