| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4470753 | 5c | EC50 | = | 8 | nM | ALA4307144 | 8.10 | nM | Homo sapiens | ||
| 2. | ALA4470753 | 5c | EC50 | = | 5 | nM | ALA4307145 | 8.30 | nM | Homo sapiens | ||
| 3. | ALA4470753 | 5c | EC50 | = | 2939 | nM | ALA4307146 | 5.53 | nM | Homo sapiens | ||
| 4. | ALA4470753 | 5c | Activity | = | 92 | % | ALA4307147 | % | Homo sapiens | |||
| 5. | ALA4470753 | 5c | Activity | = | 79 | % | ALA4307148 | % | Homo sapiens | |||
| 6. | ALA4470753 | 5c | Activity | = | 110 | % | ALA4307149 | % | Homo sapiens | |||
| 7. | ALA4470753 | 5c | Ratio EC50 | = | 367 | ALA4307150 | ||||||
| 8. | ALA4470753 | 5c | Ratio EC50 | = | 588 | ALA4307151 | Homo sapiens | |||||
| 9. | ALA4470753 | 5c | Ratio EC50 | = | 8 | ALA4307152 | Homo sapiens | |||||
| 10. | ALA4470753 | 5c | CLH | < | 9.6 | ml/min.kg | ALA4307153 | mL.min-1.kg-1 | ||||
| 11. | ALA4470753 | 5c | CLH | < | 9.6 | ml/min.kg | ALA4307154 | mL.min-1.kg-1 | ||||
| 12. | ALA4470753 | 5c | Stability | = | 88 | % | ALA4307155 | % | ||||
| 13. | ALA4470753 | 5c | Stability | = | 96 | % | ALA4307156 | % | ||||
| 14. | ALA4470753 | 5c | PPB | > | 99.99 | % | ALA4307157 | % | ||||
| 15. | ALA4470753 | 5c | PPB | > | 99.99 | % | ALA4307158 | % | ||||
| 16. | ALA4470753 | 5c | Papp | = | 0.5 | 10'-6 cm/s | ALA4307159 | 10'-6 cm/s | ||||
| 17. | ALA4470753 | 5c | Papp | = | 0.2 | 10'-6 cm/s | ALA4307160 | 10'-6 cm/s | ||||
| 18. | ALA4470753 | 5c | Ratio | = | 0.4 | ALA4307161 | ||||||
| 19. | ALA4470753 | 5c | IC50 | = | 10 | uM | ALA4307162 | 5.00 | nM | Homo sapiens | ||
| 20. | ALA4470753 | 5c | IC50 | = | 20 | uM | ALA4307163 | 4.70 | nM | Homo sapiens |
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