# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PDK4-IN-1 hydrochloride | 8c | Activity | = | 19.2 | % | ALA4333169 | % | Homo sapiens | |||
2. | PDK4-IN-1 hydrochloride | 8c | Activity | = | 5.2 | % | ALA4333168 | % | Homo sapiens | |||
3. | PDK4-IN-1 hydrochloride | 8c | Activity | = | 8.2 | % | ALA4333167 | % | Homo sapiens | |||
4. | PDK4-IN-1 hydrochloride | 8c | Activity | = | 67.4 | % | ALA4333166 | % | Homo sapiens | |||
5. | PDK4-IN-1 hydrochloride | 8c | Activity | = | 2.8 | % | ALA4333165 | % | Homo sapiens | |||
6. | PDK4-IN-1 hydrochloride | 8c | Activity | = | 2.7 | % | ALA4333164 | % | Homo sapiens | |||
7. | PDK4-IN-1 hydrochloride | 8c | Activity | = | 3.4 | % | ALA4333163 | % | Homo sapiens | |||
8. | PDK4-IN-1 hydrochloride | 8c | Activity | = | 91.1 | % | ALA4333162 | % | Homo sapiens | |||
9. | PDK4-IN-1 hydrochloride | 8c | Activity | = | 21.6 | % | ALA4333161 | % | Homo sapiens | |||
10. | PDK4-IN-1 hydrochloride | 8c | INH | = | 50.12 | % | ALA4333047 | % | Homo sapiens | |||
11. | PDK4-IN-1 hydrochloride | 8c | IC50 | = | 84 | nM | ALA4333048 | 7.08 | nM | Homo sapiens | ||
12. | PDK4-IN-1 hydrochloride | 8c | FC | = | 0.04 | ALA4333049 | Homo sapiens | |||||
13. | PDK4-IN-1 hydrochloride | 8c | FC | = | 0.18 | ALA4333050 | Homo sapiens | |||||
14. | PDK4-IN-1 hydrochloride | 8c | FC | = | 0.26 | ALA4333051 | Homo sapiens | |||||
15. | PDK4-IN-1 hydrochloride | 8c | t1/2 | > | 60 | min | ALA4333055 | hr | ||||
16. | PDK4-IN-1 hydrochloride | 8c | Drug metabolism | 0 | ALA4333056 | Metabolite_Detected | ||||||
17. | PDK4-IN-1 hydrochloride | 8c | Stability | = | 67.8 | % | ALA4333057 | % | ||||
18. | PDK4-IN-1 hydrochloride | 8c | IC50 | = | 16.3 | uM | ALA4333059 | 4.79 | nM | Homo sapiens | ||
19. | PDK4-IN-1 hydrochloride | 8c | IC50 | > | 50 | uM | ALA4333060 | nM | Homo sapiens | |||
20. | PDK4-IN-1 hydrochloride | 8c | IC50 | = | 42.4 | uM | ALA4333061 | 4.37 | nM | Homo sapiens |