# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4471658 | 5c | Retention_time | = | 9.004 | min | ALA4409103 | min | ||||
2. | ALA4471658 | 5c | Activity | 0 | ALA4409102 | Active | Homo sapiens | |||||
3. | ALA4471658 | 5c | Activity | 0 | ALA4409101 | Active | Homo sapiens | |||||
4. | ALA4471658 | 5c | Activity | 0 | ALA4409100 | Non-Toxic | Homo sapiens | |||||
5. | ALA4471658 | 5c | t1/2 | = | 24.39 | min | ALA4409099 | hr | ||||
6. | ALA4471658 | 5c | CLH | = | 47.36 | microL/min/mg | ALA4409098 | mL.min-1.g-1 | ||||
7. | ALA4471658 | 5c | K | = | 0.028 | 10'-1/min | ALA4409097 | 10'-1/min | ||||
8. | ALA4471658 | 5c | t1/2 | = | 19.91 | min | ALA4409096 | hr | ||||
9. | ALA4471658 | 5c | CLH | = | 59.22 | microL/min/mg | ALA4409095 | mL.min-1.g-1 | ||||
10. | ALA4471658 | 5c | K | = | 0.035 | 10'-1/min | ALA4409094 | 10'-1/min | ||||
11. | ALA4471658 | 5c | IC50 | = | 23 | uM | ALA4409089 | 4.64 | nM | Homo sapiens | ||
12. | ALA4471658 | 5c | IC50 | = | 68 | uM | ALA4409088 | 4.17 | nM | Mus musculus | ||
13. | ALA4471658 | 5c | Stability | = | 99.9 | % | ALA4409087 | % | ||||
14. | ALA4471658 | 5c | solubility | = | 2 | uM | ALA4409086 | nM | ||||
15. | ALA4471658 | 5c | solubility | = | 991 | uM | ALA4409085 | nM | ||||
16. | ALA4471658 | 5c | INH | 0 | ALA4409084 | Not Active | % | Mus musculus | ||||
17. | ALA4471658 | 5c | INH | 0 | ALA4409083 | Not Active | % | Mus musculus | ||||
18. | ALA4471658 | 5c | INH | 0 | ALA4409082 | Not Active | % | Mus musculus | ||||
19. | ALA4471658 | 5c | pIC50 | > | 7 | ALA4409081 | nM | Homo sapiens | ||||
20. | ALA4471658 | 5c | IC50 | < | 0.1 | uM | ALA4409081 | nM | Homo sapiens |