| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4472718 | 9 | Vdss | = | 30.3 | L/Kg | ALA4413831 | L.kg-1 | ||||
| 2. | ALA4472718 | 9 | beta t1/2 | = | 2.5 | hr | ALA4413830 | hr | ||||
| 3. | ALA4472718 | 9 | Tmax | = | 2.8 | hr | ALA4413829 | hr | ||||
| 4. | ALA4472718 | 9 | CL | = | 139 | ml/min.kg | ALA4413828 | mL.min-1.kg-1 | ||||
| 5. | ALA4472718 | 9 | Cmax | = | 0.08 | uM | ALA4413827 | nM | ||||
| 6. | ALA4472718 | 9 | F | = | 18.3 | % | ALA4413826 | % | ||||
| 7. | ALA4472718 | 9 | AUC | = | 0.66 | uM.hr | ALA4413825 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 8. | ALA4472718 | 9 | AUC | = | 0.29 | uM.hr | ALA4413824 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 9. | ALA4472718 | 9 | AUC | = | 0.45 | uM.hr | ALA4413823 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 10. | ALA4472718 | 9 | AUC | = | 0.28 | uM.hr | ALA4413822 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 11. | ALA4472718 | 9 | IC50 | = | 18.9 | uM | ALA4413821 | 4.72 | nM | Homo sapiens | ||
| 12. | ALA4472718 | 9 | Peff | = | 4.84 | 10'-6 cm/s | ALA4413820 | 10'-6 cm/s | ||||
| 13. | ALA4472718 | 9 | Stability | = | 47.6 | % | ALA4413819 | % | ||||
| 14. | ALA4472718 | 9 | Stability | = | 65.7 | % | ALA4413818 | % | ||||
| 15. | ALA4472718 | 9 | Stability | 0 | ALA4413817 | Not Determined | % | |||||
| 16. | ALA4472718 | 9 | Stability | = | 79.2 | % | ALA4413816 | % | ||||
| 17. | ALA4472718 | 9 | INH | = | 29.1 | % | ALA4413815 | % | Homo sapiens | |||
| 18. | ALA4472718 | 9 | INH | = | 31.8 | % | ALA4413814 | % | Homo sapiens | |||
| 19. | ALA4472718 | 9 | INH | = | 27.2 | % | ALA4413813 | % | Homo sapiens | |||
| 20. | ALA4472718 | 9 | INH | = | 37.7 | % | ALA4413812 | % | Homo sapiens |
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