# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4472933 | 067; 2 | AUClast | = | 126.5 | hr.ng/ml | ALA4422067 | ng.hr.mL-1 | ||||
2. | ALA4472933 | 067; 2 | Cp | = | 11.4 | ng/ml | ALA4422066 | ng/ml | ||||
3. | ALA4472933 | 067; 2 | Cp | = | 13.3 | ng/ml | ALA4422065 | ng/ml | ||||
4. | ALA4472933 | 067; 2 | Cp | = | 10.6 | ng/ml | ALA4422064 | ng/ml | ||||
5. | ALA4472933 | 067; 2 | Cp | = | 50.8 | ng/ml | ALA4422063 | ng/ml | ||||
6. | ALA4472933 | 067; 2 | AUClast | = | 691.6 | hr.ng/ml | ALA4422062 | ng.hr.mL-1 | ||||
7. | ALA4472933 | 067; 2 | Cp | = | 33.7 | ng/ml | ALA4422061 | ng/ml | ||||
8. | ALA4472933 | 067; 2 | Cp | = | 33.4 | ng/ml | ALA4422060 | ng/ml | ||||
9. | ALA4472933 | 067; 2 | Cp | = | 79.6 | ng/ml | ALA4422059 | ng/ml | ||||
10. | ALA4472933 | 067; 2 | Cp | = | 301 | ng/ml | ALA4422058 | ng/ml | ||||
11. | ALA4472933 | 067; 2 | t1/2 | = | 30 | min | ALA4422057 | hr | ||||
12. | ALA4472933 | 067; 2 | t1/2 | < | 1 | hr | ALA4422056 | hr | ||||
13. | ALA4472933 | 067; 2 | INH | 0 | ALA4422047 | Active | % | Homo sapiens | ||||
14. | ALA4472933 | 067; 2 | INH | 0 | ALA4422046 | Active | % | Homo sapiens | ||||
15. | ALA4472933 | 067; 2 | IC50 | = | 1.2 | uM | ALA4422045 | 5.92 | nM | Homo sapiens |