# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4473988 | 4 | Tmax | = | 1.6 | hr | ALA4416899 | hr | ||||
2. | ALA4473988 | 4 | Drug metabolism | = | 1.5 | % | ALA4416926 | % | Homo sapiens | |||
3. | ALA4473988 | 4 | Drug metabolism | = | 1.5 | % | ALA4416924 | % | Homo sapiens | |||
4. | ALA4473988 | 4 | beta t1/2 | = | 9.6 | hr | ALA4416929 | hr | ||||
5. | ALA4473988 | 4 | F | = | 100 | % | ALA4416928 | % | ||||
6. | ALA4473988 | 4 | Drug metabolism | 0 | ALA4416925 | Metabolite_Notdetected | Homo sapiens | |||||
7. | ALA4473988 | 4 | Drug metabolism | 0 | ALA4416927 | Metabolite_Notdetected | Homo sapiens | |||||
8. | ALA4473988 | 4 | INH | 0 | ALA4416900 | Not Active | % | Homo sapiens | ||||
9. | ALA4473988 | 4 | Ratio | = | 0.6 | ALA4416923 | ||||||
10. | ALA4473988 | 4 | Papp | = | 15.8 | 10'-6 cm/s | ALA4416922 | 10'-6 cm/s | ||||
11. | ALA4473988 | 4 | Papp | = | 28.2 | 10'-6 cm/s | ALA4416921 | 10'-6 cm/s | ||||
12. | ALA4473988 | 4 | IC50 | > | 50 | uM | ALA4416920 | nM | Homo sapiens | |||
13. | ALA4473988 | 4 | IC50 | > | 50 | uM | ALA4416919 | nM | Homo sapiens | |||
14. | ALA4473988 | 4 | IC50 | = | 46.2 | uM | ALA4416918 | 4.33 | nM | Homo sapiens | ||
15. | ALA4473988 | 4 | IC50 | > | 50 | uM | ALA4416917 | nM | Homo sapiens | |||
16. | ALA4473988 | 4 | IC50 | > | 50 | uM | ALA4416916 | nM | Homo sapiens | |||
17. | ALA4473988 | 4 | IC50 | > | 50 | uM | ALA4416915 | nM | Homo sapiens | |||
18. | ALA4473988 | 4 | IC50 | > | 50 | uM | ALA4416914 | nM | Homo sapiens | |||
19. | ALA4473988 | 4 | Stability | = | 102 | % | ALA4416913 | % | ||||
20. | ALA4473988 | 4 | t1/2 | = | 349.72 | min | ALA4416912 | hr |