# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4475066 | 4h | EC50 | = | 3.6 | uM | ALA4338387 | 5.44 | nM | Trypanosoma brucei brucei | ||
2. | ALA4475066 | 4h | EC50 | = | 5.1 | uM | ALA4338386 | 5.29 | nM | Trypanosoma brucei brucei | ||
3. | ALA4475066 | 4h | K | = | 1228 | 10'3/M/min | ALA4338385 | 10'3/M/min | Homo sapiens | |||
4. | ALA4475066 | 4h | Ki | = | 1.5 | nM | ALA4338384 | 8.82 | nM | Homo sapiens | ||
5. | ALA4475066 | 4h | INH | = | 85 | % | ALA4338379 | % | Trypanosoma brucei rhodesiense | |||
6. | ALA4475066 | 4h | Ki | = | 0.001 | nM | ALA4338382 | nM | Trypanosoma brucei rhodesiense | |||
7. | ALA4475066 | 4h | Kinact | = | 0.001 | /min | ALA4338381 | /min | Trypanosoma brucei rhodesiense | |||
8. | ALA4475066 | 4h | INH | 0 | ALA4338380 | Active | % | Trypanosoma brucei rhodesiense | ||||
9. | ALA4475066 | 4h | K | = | 881100 | 10'3/M/min | ALA4338383 | 10'3/M/min | Trypanosoma brucei rhodesiense | |||
10. | ALA4475066 | 4h | Kinact | = | 0.002 | /min | ALA4338378 | /min | Homo sapiens |