| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4475753 | 29n | Vdss | = | 6.49 | L/Kg | ALA4310461 | L.kg-1 | ||||
| 2. | ALA4475753 | 29n | t1/2 | = | 14.3 | min | ALA4310460 | hr | ||||
| 3. | ALA4475753 | 29n | CL | = | 389 | ml/min.kg | ALA4310459 | mL.min-1.kg-1 | ||||
| 4. | ALA4475753 | 29n | K(p,uu,brain) | = | 0.49 | ALA4310458 | ||||||
| 5. | ALA4475753 | 29n | Kp | = | 3.41 | ALA4310457 | ||||||
| 6. | ALA4475753 | 29n | Fu | = | 0.003 | ALA4310456 | ||||||
| 7. | ALA4475753 | 29n | Fu | = | 0.01 | ALA4310455 | ||||||
| 8. | ALA4475753 | 29n | Fu | = | 0.02 | ALA4310454 | ||||||
| 9. | ALA4475753 | 29n | Emax | = | 2.6 | % | ALA4310453 | % | Rattus norvegicus | |||
| 10. | ALA4475753 | 29n | pIC50 | = | 6.5 | ALA4310452 | 6.50 | nM | Rattus norvegicus | |||
| 11. | ALA4475753 | 29n | IC50 | = | 316 | nM | ALA4310452 | 6.50 | nM | Rattus norvegicus |
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