# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4476495 | 14e; VU6019278 | IC50 | > | 10 | uM | ALA4393086 | nM | Homo sapiens | |||
2. | ALA4476495 | 14e; VU6019278 | IC50 | > | 10 | uM | ALA4393085 | nM | Homo sapiens | |||
3. | ALA4476495 | 14e; VU6019278 | IC50 | > | 10 | uM | ALA4393084 | nM | Homo sapiens | |||
4. | ALA4476495 | 14e; VU6019278 | IC50 | > | 10 | uM | ALA4393083 | nM | Homo sapiens | |||
5. | ALA4476495 | 14e; VU6019278 | IC50 | > | 10 | uM | ALA4393082 | nM | Homo sapiens | |||
6. | ALA4476495 | 14e; VU6019278 | IC50 | > | 10 | uM | ALA4393081 | nM | Homo sapiens | |||
7. | ALA4476495 | 14e; VU6019278 | IC50 | > | 10 | uM | ALA4393080 | nM | Homo sapiens | |||
8. | ALA4476495 | 14e; VU6019278 | Drug uptake(free) | = | 6 | nM | ALA4393079 | nM | ||||
9. | ALA4476495 | 14e; VU6019278 | Drug uptake | = | 456 | nM | ALA4393078 | nM | ||||
10. | ALA4476495 | 14e; VU6019278 | Fu | = | 0.013 | ALA4393077 | ||||||
11. | ALA4476495 | 14e; VU6019278 | K(p,uu,brain) | = | 0.65 | ALA4393076 | ||||||
12. | ALA4476495 | 14e; VU6019278 | Kp | = | 4.9 | ALA4393075 | ||||||
13. | ALA4476495 | 14e; VU6019278 | Fu | = | 0.1 | ALA4393074 | ||||||
14. | ALA4476495 | 14e; VU6019278 | IC50 | = | 0.57 | uM | ALA4393072 | 6.24 | nM | Rattus norvegicus | ||
15. | ALA4476495 | 14e; VU6019278 | Activity | = | 6.3 | % | ALA4393073 | % | Rattus norvegicus | |||
16. | ALA4476495 | 14e; VU6019278 | K(p,uu,brain) | = | 0.65 | ALA5106327 | ||||||
17. | ALA4476495 | 14e; VU6019278 | Kp | = | 4.9 | ALA5106326 | ||||||
18. | ALA4476495 | 14e; VU6019278 | PPB | = | 0.1 | % | ALA5106325 | % | ||||
19. | ALA4476495 | 14e; VU6019278 | Emin | = | 0 | % | ALA5106324 | % | Homo sapiens | |||
20. | ALA4476495 | 14e; VU6019278 | pIC50 | = | 5.5 | ALA5106323 | 5.50 | nM | Homo sapiens |